Fentanyl-Type Antagonist of the μ-Opioid Receptor: Important Role of Axial Chirality in the Active Conformation.
Arita H, Tanaka R, Kikukawa S, Tomizawa T, Sakata H, Funada M, Tomiyama K, Hashimoto M, Tasaka T, Tabata H, Nakamura K, Makino K, Oshitari T, Natsugari H, Takahashi H.
Arita H, et al. Among authors: hashimoto m.
J Med Chem. 2024 Jun 13. doi: 10.1021/acs.jmedchem.4c00935. Online ahead of print.
J Med Chem. 2024.
PMID: 38869493