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Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy.
J Med Chem. 2021 Apr 8;64(7):3843-3869. doi: 10.1021/acs.jmedchem.0c02023. Epub 2021 Mar 22.
J Med Chem. 2021.
PMID: 33749283
TRPA1 modulation by piperidine carboxamides suggests an evolutionarily conserved binding site and gating mechanism.
Chernov-Rogan T, Gianti E, Liu C, Villemure E, Cridland AP, Hu X, Ballini E, Lange W, Deisemann H, Li T, Ward SI, Hackos DH, Magnuson S, Safina B, Klein ML, Volgraf M, Carnevale V, Chen J.
Chernov-Rogan T, et al. Among authors: cridland ap.
Proc Natl Acad Sci U S A. 2019 Dec 17;116(51):26008-26019. doi: 10.1073/pnas.1913929116. Epub 2019 Dec 3.
Proc Natl Acad Sci U S A. 2019.
PMID: 31796582
Free PMC article.
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Optimization of sphingosine-1-phosphate-1 receptor agonists: effects of acidic, basic, and zwitterionic chemotypes on pharmacokinetic and pharmacodynamic profiles.
Skidmore J, Heer J, Johnson CN, Norton D, Redshaw S, Sweeting J, Hurst D, Cridland A, Vesey D, Wall I, Ahmed M, Rivers D, Myatt J, Giblin G, Philpott K, Kumar U, Stevens A, Bit RA, Haynes A, Taylor S, Watson R, Witherington J, Demont E, Heightman TD.
Skidmore J, et al.
J Med Chem. 2014 Dec 26;57(24):10424-42. doi: 10.1021/jm5010336. Epub 2014 Dec 15.
J Med Chem. 2014.
PMID: 25431977
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Studies on the synthesis of the ABC rings of (+/-)-hexacyclinic acid.
Clarke PA, Cridland AP, Rolla GA, Iqbal M, Bainbridge NP, Whitwood AC, Wilson C.
Clarke PA, et al. Among authors: cridland ap.
J Org Chem. 2009 Oct 16;74(20):7812-21. doi: 10.1021/jo901547k.
J Org Chem. 2009.
PMID: 19813768
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A racemic synthesis of an AB-ring system of hexacyclinic acid.
Clarke PA, Cridland AP.
Clarke PA, et al. Among authors: cridland ap.
Org Lett. 2005 Sep 15;7(19):4221-4. doi: 10.1021/ol051633r.
Org Lett. 2005.
PMID: 16146392
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Novel enantioselective synthesis of 1,3-butadien-2-ylmethanols via tandem alkylbromide-epoxide vinylations using dimethylsulfonium methylide.
Alcaraz L, Cox K, Cridland AP, Kinchin E, Morris J, Thompson SP.
Alcaraz L, et al. Among authors: cridland ap.
Org Lett. 2005 Mar 31;7(7):1399-401. doi: 10.1021/ol0502329.
Org Lett. 2005.
PMID: 15787516
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Novel conversion of 1,2-disubstituted cis-epoxides to one-carbon homologated allylic alcohols using dimethylsulfonium methylide.
Alcaraz L, Cridland A, Kinchin E.
Alcaraz L, et al.
Org Lett. 2001 Dec 13;3(25):4051-3. doi: 10.1021/ol016782y.
Org Lett. 2001.
PMID: 11735582
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