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A Continuous Flow Process for LSN647712 via Double Organometallic Additions to Dimethylcarbamyl Chloride.
J Org Chem. 2022 Feb 18;87(4):2045-2054. doi: 10.1021/acs.joc.1c01354. Epub 2021 Aug 10.
J Org Chem. 2022.
PMID: 34374277
Discovery of Proteolysis-Targeting Chimera Molecules that Selectively Degrade the IRAK3 Pseudokinase.
Degorce SL, Tavana O, Banks E, Crafter C, Gingipalli L, Kouvchinov D, Mao Y, Pachl F, Solanki A, Valge-Archer V, Yang B, Edmondson SD.
Degorce SL, et al. Among authors: kouvchinov d.
J Med Chem. 2020 Sep 24;63(18):10460-10473. doi: 10.1021/acs.jmedchem.0c01125. Epub 2020 Sep 14.
J Med Chem. 2020.
PMID: 32803978
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Optimization of First-in-Class Dual-Acting FFAR1/FFAR4 Allosteric Modulators with Novel Mode of Action.
Lückmann M, Shenol A, Nissen TAD, Petersen JE, Kouvchinov D, Schwartz TW, Frimurer TM.
Lückmann M, et al. Among authors: kouvchinov d.
ACS Med Chem Lett. 2022 Nov 2;13(12):1839-1847. doi: 10.1021/acsmedchemlett.2c00160. eCollection 2022 Dec 8.
ACS Med Chem Lett. 2022.
PMID: 36518697
Free PMC article.
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