Search Page
Save citations to file
Email citations
Send citations to clipboard
Add to Collections
Add to My Bibliography
Create a file for external citation management software
Your saved search
Your RSS Feed
Search Results
8 results
Filters applied: . Clear all
Results are displayed in a computed author sort order.
The Results By Year timeline is not available.
Page 1
Neurosteroids and steroid hormones are allosteric modulators of muscarinic receptors.
Neuropharmacology. 2021 Nov 1;199:108798. doi: 10.1016/j.neuropharm.2021.108798. Epub 2021 Sep 22.
Neuropharmacology. 2021.
PMID: 34555368
Free article.
Neuroactive steroids, WIN-compounds and cholesterol share a common binding site on muscarinic acetylcholine receptors.
Dolejší E, Chetverikov N, Szánti-Pintér E, Nelic D, Randáková A, Doležal V, El-Fakahany EE, Kudová E, Jakubík J.
Dolejší E, et al. Among authors: nelic d.
Biochem Pharmacol. 2021 Oct;192:114699. doi: 10.1016/j.bcp.2021.114699. Epub 2021 Jul 26.
Biochem Pharmacol. 2021.
PMID: 34324870
Free article.
Item in Clipboard
Novel M2 -selective, Gi -biased agonists of muscarinic acetylcholine receptors.
Randáková A, Nelic D, Ungerová D, Nwokoye P, Su Q, Doležal V, El-Fakahany EE, Boulos J, Jakubík J.
Randáková A, et al. Among authors: nelic d.
Br J Pharmacol. 2020 May;177(9):2073-2089. doi: 10.1111/bph.14970. Epub 2020 Feb 15.
Br J Pharmacol. 2020.
PMID: 31910288
Free PMC article.
Item in Clipboard
Agonist-Specific Conformations of the M2 Muscarinic Acetylcholine Receptor Assessed by Molecular Dynamics.
Randáková A, Nelic D, Doležal V, El-Fakahany EE, Boulos J, Jakubík J.
Randáková A, et al. Among authors: nelic d.
J Chem Inf Model. 2020 Apr 27;60(4):2325-2338. doi: 10.1021/acs.jcim.0c00041. Epub 2020 Mar 13.
J Chem Inf Model. 2020.
PMID: 32130001
Item in Clipboard
Fusion with Promiscuous Gα16 Subunit Reveals Signaling Bias at Muscarinic Receptors.
Randáková A, Nelic D, Hochmalová M, Zimčík P, Mulenga MJ, Boulos J, Jakubík J.
Randáková A, et al. Among authors: nelic d.
Int J Mol Sci. 2021 Sep 18;22(18):10089. doi: 10.3390/ijms221810089.
Int J Mol Sci. 2021.
PMID: 34576254
Free PMC article.
Item in Clipboard
Guanidine Derivatives: How Simple Structural Modification of Histamine H3R Antagonists Has Led to the Discovery of Potent Muscarinic M2R/M4R Antagonists.
Staszewski M, Nelic D, Jończyk J, Dubiel M, Frank A, Stark H, Bajda M, Jakubik J, Walczyński K.
Staszewski M, et al. Among authors: nelic d.
ACS Chem Neurosci. 2021 Jul 7;12(13):2503-2519. doi: 10.1021/acschemneuro.1c00237. Epub 2021 Jun 8.
ACS Chem Neurosci. 2021.
PMID: 34100603
Free PMC article.
Item in Clipboard
Agonist-selective activation of individual G-proteins by muscarinic receptors.
Nelic D, Chetverikov N, Hochmalová M, Diaz C, Doležal V, Boulos J, Jakubík J, Martemyanov K, Janoušková-Randáková A.
Nelic D, et al.
Sci Rep. 2024 Apr 26;14(1):9652. doi: 10.1038/s41598-024-60259-4.
Sci Rep. 2024.
PMID: 38671143
Free PMC article.
Item in Clipboard
A critical re-evaluation of the slope factor of the operational model of agonism: When to exponentiate operational efficacy.
Randáková A, Nelic D, Jakubík J.
Randáková A, et al. Among authors: nelic d.
Sci Rep. 2023 Oct 16;13(1):17587. doi: 10.1038/s41598-023-45004-7.
Sci Rep. 2023.
PMID: 37845324
Free PMC article.
Item in Clipboard
Cite
Cite