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Design and discovery of C2-fluoroalkyl iminothiazine dioxides as BACE inhibitors.
Bioorg Med Chem Lett. 2022 Jan 15;56:128463. doi: 10.1016/j.bmcl.2021.128463. Epub 2021 Nov 24.
Bioorg Med Chem Lett. 2022.
PMID: 34838652
Discovery of 1-amino-5H-pyrido[4,3-b]indol-4-carboxamide inhibitors of Janus kinase 2 (JAK2) for the treatment of myeloproliferative disorders.
Lim J, Taoka B, Otte RD, Spencer K, Dinsmore CJ, Altman MD, Chan G, Rosenstein C, Sharma S, Su HP, Szewczak AA, Xu L, Yin H, Zugay-Murphy J, Marshall CG, Young JR.
Lim J, et al.
J Med Chem. 2011 Oct 27;54(20):7334-49. doi: 10.1021/jm200909u. Epub 2011 Sep 26.
J Med Chem. 2011.
PMID: 21942426
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Efficacious intermittent dosing of a novel JAK2 inhibitor in mouse models of polycythemia vera.
Kraus M, Wang Y, Aleksandrowicz D, Bachman E, Szewczak AA, Walker D, Xu L, Bouthillette M, Childers KM, Dolinski B, Haidle AM, Kopinja J, Lee L, Lim J, Little KD, Ma Y, Mathur A, Mo JR, O'Hare E, Otte RD, Taoka BM, Wang W, Yin H, Zabierek AA, Zhang W, Zhao S, Zhu J, Young JR, Marshall CG.
Kraus M, et al. Among authors: taoka bm.
PLoS One. 2012;7(5):e37207. doi: 10.1371/journal.pone.0037207. Epub 2012 May 18.
PLoS One. 2012.
PMID: 22623993
Free PMC article.
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Small molecule glucagon receptor antagonists: an updated patent review (2015-2019).
Cheng C, Jabri S, Taoka BM, Sinz CJ.
Cheng C, et al. Among authors: taoka bm.
Expert Opin Ther Pat. 2020 Jul;30(7):509-526. doi: 10.1080/13543776.2020.1769600. Epub 2020 Jun 18.
Expert Opin Ther Pat. 2020.
PMID: 32552241
Review.
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Asymmetric Mannich reactions of beta-keto esters with acyl imines catalyzed by cinchona alkaloids.
Lou S, Taoka BM, Ting A, Schaus SE.
Lou S, et al. Among authors: taoka bm.
J Am Chem Soc. 2005 Aug 17;127(32):11256-7. doi: 10.1021/ja0537373.
J Am Chem Soc. 2005.
PMID: 16089450
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