Discovery of JNJ-74856665: A Novel Isoquinolinone DHODH Inhibitor for the Treatment of AML.
DeRatt LG, Zhang Z, Pietsch C, Cisar JS, Zhang X, Wang W, Tanner A, Matico R, Shaffer P, Jacoby E, Kazmi F, Shukla N, Bush TL, Patrick A, Philippar U, Attar R, Edwards JP, Kuduk SD.
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J Med Chem. 2024 Jun 18. doi: 10.1021/acs.jmedchem.4c00809. Online ahead of print.
J Med Chem. 2024.
PMID: 38889244