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Absorption, distribution, metabolism and excretion of 14C-vatiquinone in rats, dogs, and human subjects.
Xenobiotica. 2023 May;53(5):396-411. doi: 10.1080/00498254.2023.2245459. Epub 2023 Aug 18.
Xenobiotica. 2023.
PMID: 37552765
First-in-Human Studies of Pharmacokinetics and Safety of Utreloxastat (PTC857), a Novel 15-Lipooxygenase Inhibitor for the Treatment of Amyotrophic Lateral Sclerosis.
Gao L, Giannousis P, Thoolen M, Kaushik D, Latham J, Tansy A, Ma J, Johnston M, Dali M, Golden L, Klein M, Kong R, Trimmer J.
Gao L, et al. Among authors: giannousis p.
Clin Pharmacol Drug Dev. 2023 Feb;12(2):141-151. doi: 10.1002/cpdd.1203. Epub 2022 Dec 14.
Clin Pharmacol Drug Dev. 2023.
PMID: 36516010
Free PMC article.
Clinical Trial.
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The First Enantioselective Synthesis of (2R,2'R)-threo-(+)-Methylphenidate Hydrochloride.
Prashad M, Kim HY, Lu Y, Liu Y, Har D, Repic O, Blacklock TJ, Giannousis P.
Prashad M, et al. Among authors: giannousis p.
J Org Chem. 1999 Mar 5;64(5):1750-1753. doi: 10.1021/jo9821473.
J Org Chem. 1999.
PMID: 11674251
No abstract available.
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Phosphorus amino acid analogues as inhibitors of leucine aminopeptidase.
Giannousis PP, Bartlett PA.
Giannousis PP, et al.
J Med Chem. 1987 Sep;30(9):1603-9. doi: 10.1021/jm00392a014.
J Med Chem. 1987.
PMID: 3625708
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Phosphorus-containing peptide analogs as peptidase inhibitors.
Bartlett PA, Marlowe CK, Giannousis PP, Hanson JE.
Bartlett PA, et al. Among authors: giannousis pp.
Cold Spring Harb Symp Quant Biol. 1987;52:83-90. doi: 10.1101/sqb.1987.052.01.012.
Cold Spring Harb Symp Quant Biol. 1987.
PMID: 2841072
No abstract available.
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Geometric specificity of alcohol dehydrogenases and its potential for separation of trans and cis isomers of unsaturated aldehydes.
Klibanov AM, Giannousis PP.
Klibanov AM, et al. Among authors: giannousis pp.
Proc Natl Acad Sci U S A. 1982 Jun;79(11):3462-5. doi: 10.1073/pnas.79.11.3462.
Proc Natl Acad Sci U S A. 1982.
PMID: 7048306
Free PMC article.
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