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Liver-Selective Imidazolopyrazine Mitochondrial Uncoupler SHD865 Reverses Adiposity and Glucose Intolerance in Mice.
Diabetes. 2024 Mar 1;73(3):374-384. doi: 10.2337/db23-0233.
Diabetes. 2024.
PMID: 37870907
Free PMC article.
Conversion of oxadiazolo[3,4-b]pyrazines to imidazo[4,5-b]pyrazines via a tandem reduction-cyclization sequence generates new mitochondrial uncouplers.
Dai Y, Santiago-Rivera JA, Hargett S, Salamoun JM, Hoehn KL, Santos WL.
Dai Y, et al. Among authors: santiago rivera ja.
Bioorg Med Chem Lett. 2022 Oct 1;73:128912. doi: 10.1016/j.bmcl.2022.128912. Epub 2022 Jul 28.
Bioorg Med Chem Lett. 2022.
PMID: 35907607
Free PMC article.
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