Emmitte KA - Search Results

1

Structure-Activity Relationship Studies in a Series of Xanthine Inhibitors of SLACK Potassium Channels.

Qunies AM, Spitznagel BD, Du Y, Peprah PK, Mohamed YK, Weaver CD, Emmitte KA. Qunies AM, et al. Among authors: emmitte ka. Molecules. 2024 May 22;29(11):2437. doi: 10.3390/molecules29112437. Molecules. 2024. PMID: 38893312 Free PMC article.

2

Quercetin and Related Analogs as Therapeutics to Promote Tissue Repair.

McKay TB, Emmitte KA, German C, Karamichos D. McKay TB, et al. Among authors: emmitte ka. Bioengineering (Basel). 2023 Sep 25;10(10):1127. doi: 10.3390/bioengineering10101127. Bioengineering (Basel). 2023. PMID: 37892857 Free PMC article. Review.

3

Heterozygous expression of a Kcnt1 gain-of-function variant has differential effects on SST- and PV-expressing cortical GABAergic neurons.

Shore AN, Li K, Safari M, Qunies AM, Spitznagel BD, Weaver CD, Emmitte KA, Frankel WN, Weston MC. Shore AN, et al. Among authors: emmitte ka. bioRxiv [Preprint]. 2024 May 29:2023.10.11.561953. doi: 10.1101/2023.10.11.561953. bioRxiv. 2024. PMID: 37873369 Free PMC article. Preprint.

4

Design, synthesis, and biological evaluation of a novel series of 1,2,4-oxadiazole inhibitors of SLACK potassium channels: Identification of in vitro tool VU0935685.

Qunies AM, Spitznagel BD, Du Y, David Weaver C, Emmitte KA. Qunies AM, et al. Among authors: emmitte ka. Bioorg Med Chem. 2023 Nov 15;95:117487. doi: 10.1016/j.bmc.2023.117487. Epub 2023 Sep 30. Bioorg Med Chem. 2023. PMID: 37812884

5

Structure-Activity Relationship Study of the High-Affinity Neuropeptide Y₄ Receptor Positive Allosteric Modulator VU0506013.

Schüß C, Vu O, Mishra NM, Tough IR, Du Y, Stichel J, Cox HM, Weaver CD, Meiler J, Emmitte KA, Beck-Sickinger AG. Schüß C, et al. Among authors: emmitte ka. J Med Chem. 2023 Jul 13;66(13):8745-8766. doi: 10.1021/acs.jmedchem.3c00383. Epub 2023 Jun 20. J Med Chem. 2023. PMID: 37339079

6

Structure-activity relationship studies in a new series of 2-amino-N-phenylacetamide inhibitors of Slack potassium channels.

Qunies AM, Mishra NM, Spitznagel BD, Du Y, Acuña VS, David Weaver C, Emmitte KA. Qunies AM, et al. Among authors: emmitte ka. Bioorg Med Chem Lett. 2022 Nov 15;76:129013. doi: 10.1016/j.bmcl.2022.129013. Epub 2022 Sep 29. Bioorg Med Chem Lett. 2022. PMID: 36184030 Free PMC article.

7

Negative allosteric modulators of group II metabotropic glutamate receptors: A patent review (2015 - present).

Qunies AM, Emmitte KA. Qunies AM, et al. Among authors: emmitte ka. Expert Opin Ther Pat. 2021 Aug;31(8):687-708. doi: 10.1080/13543776.2021.1903431. Epub 2021 Mar 31. Expert Opin Ther Pat. 2021. PMID: 33719801 Review.

8

Highly Selective Y₄ Receptor Antagonist Binds in an Allosteric Binding Pocket.

Schüß C, Vu O, Schubert M, Du Y, Mishra NM, Tough IR, Stichel J, Weaver CD, Emmitte KA, Cox HM, Meiler J, Beck-Sickinger AG. Schüß C, et al. Among authors: emmitte ka. J Med Chem. 2021 Mar 11;64(5):2801-2814. doi: 10.1021/acs.jmedchem.0c02000. Epub 2021 Feb 17. J Med Chem. 2021. PMID: 33595306

9

VU0606170, a Selective Slack Channels Inhibitor, Decreases Calcium Oscillations in Cultured Cortical Neurons.

Spitznagel BD, Mishra NM, Qunies AM, Prael FJ 3rd, Du Y, Kozek KA, Lazarenko RM, Denton JS, Emmitte KA, Weaver CD. Spitznagel BD, et al. Among authors: emmitte ka. ACS Chem Neurosci. 2020 Nov 4;11(21):3658-3671. doi: 10.1021/acschemneuro.0c00583. Epub 2020 Oct 14. ACS Chem Neurosci. 2020. PMID: 33143429

10

Discovery of VU2957 (Valiglurax): An mGlu₄ Positive Allosteric Modulator Evaluated as a Preclinical Candidate for the Treatment of Parkinson's Disease.

Panarese JD, Engers DW, Wu YJ, Bronson JJ, Macor JE, Chun A, Rodriguez AL, Felts AS, Engers JL, Loch MT, Emmitte KA, Castelhano AL, Kates MJ, Nader MA, Jones CK, Blobaum AL, Conn PJ, Niswender CM, Hopkins CR, Lindsley CW. Panarese JD, et al. Among authors: emmitte ka. ACS Med Chem Lett. 2018 Oct 16;10(3):255-260. doi: 10.1021/acsmedchemlett.8b00426. eCollection 2019 Mar 14. ACS Med Chem Lett. 2018. PMID: 30891122 Free PMC article.

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