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Synthesis and Profiling of a Novel Potent Selective Inhibitor of CHK1 Kinase Possessing Unusual N-trifluoromethylpyrazole Pharmacophore Resistant to Metabolic N-dealkylation.
Samadder P, Suchánková T, Hylse O, Khirsariya P, Nikulenkov F, Drápela S, Straková N, Vaňhara P, Vašíčková K, Kolářová H, Binó L, Bittová M, Ovesná P, Kollár P, Fedr R, Ešner M, Jaroš J, Hampl A, Krejčí L, Paruch K, Souček K. Samadder P, et al. Among authors: ovesna p. Mol Cancer Ther. 2017 Sep;16(9):1831-1842. doi: 10.1158/1535-7163.MCT-17-0018. Epub 2017 Jun 15. Mol Cancer Ther. 2017. PMID: 28619751
Casein kinase 1 is a therapeutic target in chronic lymphocytic leukemia.
Janovska P, Verner J, Kohoutek J, Bryjova L, Gregorova M, Dzimkova M, Skabrahova H, Radaszkiewicz T, Ovesna P, Vondalova Blanarova O, Nemcova T, Hoferova Z, Vasickova K, Smyckova L, Egle A, Pavlova S, Poppova L, Plevova K, Pospisilova S, Bryja V. Janovska P, et al. Among authors: ovesna p. Blood. 2018 Mar 15;131(11):1206-1218. doi: 10.1182/blood-2017-05-786947. Epub 2018 Jan 9. Blood. 2018. PMID: 29317454 Free article.
Single-cell protein profiling defines cell populations associated with triple-negative breast cancer aggressiveness.
Kvokačková B, Fedr R, Kužílková D, Stuchlý J, Vávrová A, Navrátil J, Fabian P, Ondruššek R, Ovesná P, Remšík J, Bouchal J, Kalina T, Souček K. Kvokačková B, et al. Among authors: ovesna p. Mol Oncol. 2023 Jun;17(6):1024-1040. doi: 10.1002/1878-0261.13365. Epub 2023 Jan 25. Mol Oncol. 2023. PMID: 36550781 Free PMC article.
Orthotopic model for the analysis of melanoma circulating tumor cells.
Pícková M, Kahounová Z, Radaszkiewicz T, Procházková J, Fedr R, Nosková M, Radaszkiewicz KA, Ovesná P, Bryja V, Souček K. Pícková M, et al. Among authors: ovesna p. Sci Rep. 2024 Apr 3;14(1):7827. doi: 10.1038/s41598-024-58236-y. Sci Rep. 2024. PMID: 38570556 Free PMC article.
WNT signaling inducing activity in ascites predicts poor outcome in ovarian cancer.
Kotrbová A, Ovesná P, Gybel' T, Radaszkiewicz T, Bednaříková M, Hausnerová J, Jandáková E, Minář L, Crha I, Weinberger V, Záveský L, Bryja V, Pospíchalová V. Kotrbová A, et al. Among authors: ovesna p. Theranostics. 2020 Jan 1;10(2):537-552. doi: 10.7150/thno.37423. eCollection 2020. Theranostics. 2020. PMID: 31903136 Free PMC article.
Specific alterations of sphingolipid metabolism identified in EpCAM-positive cells isolated from human colon tumors.
Procházková J, Slavík J, Bouchal J, Levková M, Hušková Z, Ehrmann J, Ovesná P, Kolář Z, Skalický P, Straková N, Zapletal O, Kozubík A, Hofmanová J, Vondráček J, Machala M. Procházková J, et al. Among authors: ovesna p. Biochim Biophys Acta Mol Cell Biol Lipids. 2020 Sep;1865(9):158742. doi: 10.1016/j.bbalip.2020.158742. Epub 2020 May 21. Biochim Biophys Acta Mol Cell Biol Lipids. 2020. PMID: 32447053 No abstract available.
Microenvironmental interactions between endothelial and lymphoma cells: a role for the canonical WNT pathway in Hodgkin lymphoma.
Linke F, Harenberg M, Nietert MM, Zaunig S, von Bonin F, Arlt A, Szczepanowski M, Weich HA, Lutz S, Dullin C, Janovská P, Krafčíková M, Trantírek L, Ovesná P, Klapper W, Beissbarth T, Alves F, Bryja V, Trümper L, Wilting J, Kube D. Linke F, et al. Among authors: ovesna p. Leukemia. 2017 Feb;31(2):361-372. doi: 10.1038/leu.2016.232. Epub 2016 Aug 18. Leukemia. 2017. PMID: 27535218
72 results