Pockes S - Search Results

1

Initial Characterization of a Transgenic Mouse with Overexpression of the Human H₁-Histamine Receptor on the Heart.

Rayo Abella LM, Jacob H, Keller M, Schindler L, Pockes S, Pitzl S, Klimas J, Hadova K, Schneider S, Buchwalow IB, Jin C, Panula P, Kirchhefer U, Neumann J, Gergs U. Rayo Abella LM, et al. Among authors: pockes s. J Pharmacol Exp Ther. 2024 Apr 18;389(2):174-185. doi: 10.1124/jpet.123.002060. J Pharmacol Exp Ther. 2024. PMID: 38531640

2

Activation of Multiple G Protein Pathways to Characterize the Five Dopamine Receptor Subtypes Using Bioluminescence Technology.

Mönnich D, Humphrys LJ, Höring C, Hoare BL, Forster L, Pockes S. Mönnich D, et al. Among authors: pockes s. ACS Pharmacol Transl Sci. 2024 Feb 6;7(3):834-854. doi: 10.1021/acsptsci.3c00339. eCollection 2024 Mar 8. ACS Pharmacol Transl Sci. 2024. PMID: 38481695

3

Cryo-EM structure of cell-free synthesized human histamine 2 receptor/G_s complex in nanodisc environment.

Köck Z, Schnelle K, Persechino M, Umbach S, Schihada H, Januliene D, Parey K, Pockes S, Kolb P, Dötsch V, Möller A, Hilger D, Bernhard F. Köck Z, et al. Among authors: pockes s. Nat Commun. 2024 Feb 28;15(1):1831. doi: 10.1038/s41467-024-46096-z. Nat Commun. 2024. PMID: 38418462 Free PMC article.

4

Shedding Light on the D₁ -Like Receptors: A Fluorescence-Based Toolbox for Visualization of the D₁ and D₅ Receptors.

Rosier N, Mönnich D, Nagl M, Schihada H, Sirbu A, Konar N, Reyes-Resina I, Navarro G, Franco R, Kolb P, Annibale P, Pockes S. Rosier N, et al. Among authors: pockes s. Chembiochem. 2024 Jan 15;25(2):e202300658. doi: 10.1002/cbic.202300658. Epub 2023 Nov 20. Chembiochem. 2024. PMID: 37983731

5

Discovery of a Tritiated Radioligand with High Affinity and Selectivity for the Histamine H₃ Receptor.

Mönnich D, Nagl M, Forster L, Rosier N, Igel P, Pockes S. Mönnich D, et al. Among authors: pockes s. ACS Med Chem Lett. 2023 Oct 17;14(11):1589-1595. doi: 10.1021/acsmedchemlett.3c00413. eCollection 2023 Nov 9. ACS Med Chem Lett. 2023. PMID: 37974943

6

Fluorescent Tools for the Imaging of Dopamine D₂ -Like Receptors.

Nagl M, Mönnich D, Rosier N, Schihada H, Sirbu A, Konar N, Reyes-Resina I, Navarro G, Franco R, Kolb P, Annibale P, Pockes S. Nagl M, et al. Among authors: pockes s. Chembiochem. 2024 Jan 15;25(2):e202300659. doi: 10.1002/cbic.202300659. Epub 2023 Nov 20. Chembiochem. 2024. PMID: 37942961

7

Development of Fluorescent AF64394 Analogues Enables Real-Time Binding Studies for the Orphan Class A GPCR GPR3.

Bresinsky M, Shahraki A, Kolb P, Pockes S, Schihada H. Bresinsky M, et al. Among authors: pockes s. J Med Chem. 2023 Nov 9;66(21):15025-15041. doi: 10.1021/acs.jmedchem.3c01707. Epub 2023 Oct 31. J Med Chem. 2023. PMID: 37907069 Free PMC article.

8

Clonidine stimulates force of contraction via histamine H₂ receptors in the human atrium.

Neumann J, Pockes S, Humphrys LJ, Mönnich D, Forster L, Kirchhefer U, Hofmann B, Gergs U. Neumann J, et al. Among authors: pockes s. Naunyn Schmiedebergs Arch Pharmacol. 2024 Jan;397(1):617-626. doi: 10.1007/s00210-023-02635-x. Epub 2023 Jul 25. Naunyn Schmiedebergs Arch Pharmacol. 2024. PMID: 37490122 Free PMC article.

9

An electrophilic fragment screening for the development of small molecules targeting caspase-2.

Cuellar ME, Yang M, Karavadhi S, Zhang YQ, Zhu H, Sun H, Shen M, Hall MD, Patnaik S, Ashe KH, Walters MA, Pockes S. Cuellar ME, et al. Among authors: pockes s. Eur J Med Chem. 2023 Nov 5;259:115632. doi: 10.1016/j.ejmech.2023.115632. Epub 2023 Jul 11. Eur J Med Chem. 2023. PMID: 37453329

10

Dual Piperidine-Based Histamine H₃ and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain.

Szczepańska K, Karcz T, Dichiara M, Mogilski S, Kalinowska-Tłuścik J, Pilarski B, Leniak A, Pietruś W, Podlewska S, Popiołek-Barczyk K, Humphrys LJ, Ruiz-Cantero MC, Reiner-Link D, Leitzbach L, Łażewska D, Pockes S, Górka M, Zmysłowski A, Calmels T, Cobos EJ, Marrazzo A, Stark H, Bojarski AJ, Amata E, Kieć-Kononowicz K. Szczepańska K, et al. Among authors: pockes s. J Med Chem. 2023 Jul 27;66(14):9658-9683. doi: 10.1021/acs.jmedchem.3c00430. Epub 2023 Jul 7. J Med Chem. 2023. PMID: 37418295 Free PMC article.

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