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Synthesis, biological activity, and molecular modeling of selective 5-HT(2C/2B) receptor antagonists.
J Med Chem. 1996 Dec 6;39(25):4966-77. doi: 10.1021/jm960571v.
J Med Chem. 1996.
PMID: 8960557
Novel and selective 5-HT2C/2B receptor antagonists as potential anxiolytic agents: synthesis, quantitative structure-activity relationships, and molecular modeling of substituted 1-(3-pyridylcarbamoyl)indolines.
Bromidge SM, Dabbs S, Davies DT, Duckworth DM, Forbes IT, Ham P, Jones GE, King FD, Saunders DV, Starr S, Thewlis KM, Wyman PA, Blaney FE, Naylor CB, Bailey F, Blackburn TP, Holland V, Kennett GA, Riley GJ, Wood MD.
Bromidge SM, et al. Among authors: saunders dv.
J Med Chem. 1998 May 7;41(10):1598-612. doi: 10.1021/jm970741j.
J Med Chem. 1998.
PMID: 9572885
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Model studies on a synthetically facile series of N-substituted phenyl-N'-pyridin-3-yl ureas leading to 1-(3-pyridylcarbamoyl) indolines that are potent and selective 5-HT(2C/2B) receptor antagonists.
Bromidge SM, Dabbs S, Davies DT, Davies S, Duckworth DM, Forbes IT, Gadre A, Ham P, Jones GE, King FD, Saunders DV, Thewlis KM, Vyas D, Blackburn TP, Holland V, Kennett GA, Riley GJ, Wood MD.
Bromidge SM, et al. Among authors: saunders dv.
Bioorg Med Chem. 1999 Dec;7(12):2767-73. doi: 10.1016/s0968-0896(99)00228-x.
Bioorg Med Chem. 1999.
PMID: 10658582
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A novel, potent, and selective 5-HT(7) antagonist: (R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolidine-1-sulfonyl) phen ol (SB-269970).
Lovell PJ, Bromidge SM, Dabbs S, Duckworth DM, Forbes IT, Jennings AJ, King FD, Middlemiss DN, Rahman SK, Saunders DV, Collin LL, Hagan JJ, Riley GJ, Thomas DR.
Lovell PJ, et al. Among authors: saunders dv.
J Med Chem. 2000 Feb 10;43(3):342-5. doi: 10.1021/jm991151j.
J Med Chem. 2000.
PMID: 10669560
No abstract available.
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Biarylcarbamoylindolines are novel and selective 5-HT(2C) receptor inverse agonists: identification of 5-methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a potential antidepressant/anxiolytic agent.
Bromidge SM, Dabbs S, Davies DT, Davies S, Duckworth DM, Forbes IT, Gaster LM, Ham P, Jones GE, King FD, Mulholland KR, Saunders DV, Wyman PA, Blaney FE, Clarke SE, Blackburn TP, Holland V, Kennett GA, Lightowler S, Middlemiss DN, Trail B, Riley GJ, Wood MD.
Bromidge SM, et al. Among authors: saunders dv.
J Med Chem. 2000 Mar 23;43(6):1123-34. doi: 10.1021/jm990388c.
J Med Chem. 2000.
PMID: 10737744
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1-[2-[(Heteroaryloxy)heteroaryl]carbamoyl]indolines: novel and selective 5-HT2C receptor inverse agonists with potential as antidepressant/anxiolytic agents.
Bromidge SM, Dabbs S, Davies S, Duckworth DM, Forbes IT, Jones GE, Jones J, King FD, Saunders DV, Blackburn TP, Holland V, Kennett GA, Lightowler S, Middlemiss DN, Riley GJ, Trail B, Wood MD.
Bromidge SM, et al. Among authors: saunders dv.
Bioorg Med Chem Lett. 2000 Aug 21;10(16):1863-6. doi: 10.1016/s0960-894x(00)00364-4.
Bioorg Med Chem Lett. 2000.
PMID: 10969986
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