Discovery of 5-(pyridin-3-yl)-1H-indole-4,7-diones as indoleamine 2,3-dioxygenase 1 (IDO1) inhibitors.
Bioorg Med Chem Lett. 2020 Feb 15;30(4):126901. doi: 10.1016/j.bmcl.2019.126901. Epub 2019 Dec 17.
Bioorg Med Chem Lett. 2020.
PMID: 31882299