Localization and substrate selectivity of sea urchin multidrug (MDR) efflux transporters.
Gökirmak T, Campanale JP, Shipp LE, Moy GW, Tao H, Hamdoun A.
Gökirmak T, et al.
J Biol Chem. 2012 Dec 21;287(52):43876-83. doi: 10.1074/jbc.M112.424879. Epub 2012 Nov 2.
J Biol Chem. 2012.
PMID: 23124201
Free PMC article.
Using this assay, we found that sea urchin MDR transporters export canonical MDR susbtrates such as calcein-AM, bodipy-verapamil, bodipy-vinblastine, and mitoxantrone. In addition, we characterized the impact of nonconservative substitutions in the primary sequences …
Using this assay, we found that sea urchin MDR transporters export canonical MDR susbtrates such as calcein-AM, bodipy-verapamil …