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Results by year
Table representation of search results timeline featuring number of search results per year.
Year | Number of Results |
---|---|
2012 | 1 |
2013 | 5 |
2014 | 1 |
2015 | 1 |
2024 | 0 |
Search Results
7 results
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Page 1
A novel quinoline derivative that inhibits mycobacterial FtsZ.
Tuberculosis (Edinb). 2013 Jul;93(4):398-400. doi: 10.1016/j.tube.2013.04.002. Epub 2013 May 4.
Tuberculosis (Edinb). 2013.
PMID: 23647650
Free PMC article.
Combining computational methods for hit to lead optimization in Mycobacterium tuberculosis drug discovery.
Ekins S, Freundlich JS, Hobrath JV, Lucile White E, Reynolds RC.
Ekins S, et al.
Pharm Res. 2014 Feb;31(2):414-35. doi: 10.1007/s11095-013-1172-7. Epub 2013 Oct 17.
Pharm Res. 2014.
PMID: 24132686
Free PMC article.
Item in Clipboard
Open Source Bayesian Models. 1. Application to ADME/Tox and Drug Discovery Datasets.
Clark AM, Dole K, Coulon-Spektor A, McNutt A, Grass G, Freundlich JS, Reynolds RC, Ekins S.
Clark AM, et al.
J Chem Inf Model. 2015 Jun 22;55(6):1231-45. doi: 10.1021/acs.jcim.5b00143. Epub 2015 Jun 3.
J Chem Inf Model. 2015.
PMID: 25994950
Free PMC article.
Item in Clipboard
Identification of novel Mt-Guab2 inhibitor series active against M. tuberculosis.
Usha V, Hobrath JV, Gurcha SS, Reynolds RC, Besra GS.
Usha V, et al.
PLoS One. 2012;7(3):e33886. doi: 10.1371/journal.pone.0033886. Epub 2012 Mar 29.
PLoS One. 2012.
PMID: 22479467
Free PMC article.
Item in Clipboard
Bayesian models leveraging bioactivity and cytotoxicity information for drug discovery.
Ekins S, Reynolds RC, Kim H, Koo MS, Ekonomidis M, Talaue M, Paget SD, Woolhiser LK, Lenaerts AJ, Bunin BA, Connell N, Freundlich JS.
Ekins S, et al.
Chem Biol. 2013 Mar 21;20(3):370-8. doi: 10.1016/j.chembiol.2013.01.011.
Chem Biol. 2013.
PMID: 23521795
Free PMC article.
Item in Clipboard
Fusing dual-event data sets for Mycobacterium tuberculosis machine learning models and their evaluation.
Ekins S, Freundlich JS, Reynolds RC.
Ekins S, et al.
J Chem Inf Model. 2013 Nov 25;53(11):3054-63. doi: 10.1021/ci400480s. Epub 2013 Oct 30.
J Chem Inf Model. 2013.
PMID: 24144044
Free PMC article.
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Enhancing hit identification in Mycobacterium tuberculosis drug discovery using validated dual-event Bayesian models.
Ekins S, Reynolds RC, Franzblau SG, Wan B, Freundlich JS, Bunin BA.
Ekins S, et al.
PLoS One. 2013 May 7;8(5):e63240. doi: 10.1371/journal.pone.0063240. Print 2013.
PLoS One. 2013.
PMID: 23667592
Free PMC article.
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