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Year | Number of Results |
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2020 | 1 |
2024 | 2 |
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Orphan GPR52 as an emerging neurotherapeutic target.
Drug Discov Today. 2024 Apr;29(4):103922. doi: 10.1016/j.drudis.2024.103922. Epub 2024 Feb 20.
Drug Discov Today. 2024.
PMID: 38387741
Review.
Discovery of Potent and Brain-Penetrant GPR52 Agonist that Suppresses Psychostimulant Behavior.
Wang P, Felsing DE, Chen H, Stutz SJ, Murphy RE, Cunningham KA, Allen JA, Zhou J.
Wang P, et al.
J Med Chem. 2020 Nov 25;63(22):13951-13972. doi: 10.1021/acs.jmedchem.0c01498. Epub 2020 Nov 16.
J Med Chem. 2020.
PMID: 33198466
Free PMC article.
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Discovery of 3-((4-Benzylpyridin-2-yl)amino)benzamides as Potent GPR52 G Protein-Biased Agonists.
Murphy RE, Wang P, Ali S, Smith HR, Felsing DE, Chen H, Zhou J, Allen JA.
Murphy RE, et al.
J Med Chem. 2024 Jun 13;67(11):9709-9730. doi: 10.1021/acs.jmedchem.4c00856. Epub 2024 May 24.
J Med Chem. 2024.
PMID: 38788241
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