Akram MS - Search Results

1

Synthesis, crystal structure determination, biological screening and docking studies of N¹-substituted derivatives of 2,3-dihydroquinazolin-4(1H)-one as inhibitors of cholinesterases.

Sultana N, Sarfraz M, Tanoli ST, Akram MS, Sadiq A, Rashid U, Tariq MI. Sultana N, et al. Among authors: akram ms. Bioorg Chem. 2017 Jun;72:256-267. doi: 10.1016/j.bioorg.2017.04.009. Epub 2017 Apr 17. Bioorg Chem. 2017. PMID: 28495556

2

Synthesis, biological evaluation and docking studies of 2,3-dihydroquinazolin-4(1H)-one derivatives as inhibitors of cholinesterases.

Sarfraz M, Sultana N, Rashid U, Akram MS, Sadiq A, Tariq MI. Sarfraz M, et al. Among authors: akram ms. Bioorg Chem. 2017 Feb;70:237-244. doi: 10.1016/j.bioorg.2017.01.004. Epub 2017 Jan 17. Bioorg Chem. 2017. PMID: 28126287 Free article.

3

Metal based drugs: design, synthesis and in-vitro antimicrobial screening of Co(II), Ni(II), Cu(II) and Zn(II) complexes with some new carboxamide derived compounds: crystal structures of N-[ethyl(propan-2-yl)carbamothioyl]thiophene-2-carboxamide and its copper(II) complex.

Sumrra SH, Hanif M, Chohan ZH, Akram MS, Akhtar J, Al-Shehri SM. Sumrra SH, et al. Among authors: akram ms. J Enzyme Inhib Med Chem. 2016 Aug;31(4):590-8. doi: 10.3109/14756366.2015.1050011. Epub 2015 Jun 11. J Enzyme Inhib Med Chem. 2016. PMID: 26067080

4

Metal-based ethanolamine-derived compounds: a note on their synthesis, characterization and bioactivity.

Amjad M, Sumrra SH, Akram MS, Chohan ZH. Amjad M, et al. Among authors: akram ms. J Enzyme Inhib Med Chem. 2016;31(sup4):88-97. doi: 10.1080/14756366.2016.1220375. Epub 2016 Aug 24. J Enzyme Inhib Med Chem. 2016. PMID: 27557038

5

Pharmacophore Modeling and in Silico/in Vitro Screening for Human Cytochrome P450 11B1 and Cytochrome P450 11B2 Inhibitors.

Akram M, Waratchareeyakul W, Haupenthal J, Hartmann RW, Schuster D. Akram M, et al. Front Chem. 2017 Dec 19;5:104. doi: 10.3389/fchem.2017.00104. eCollection 2017. Front Chem. 2017. PMID: 29312923 Free PMC article.

6

Antimicrobial metal-based thiophene derived compounds.

Yasmeen S, Sumrra SH, Akram MS, Chohan ZH. Yasmeen S, et al. Among authors: akram ms. J Enzyme Inhib Med Chem. 2017 Dec;32(1):106-112. doi: 10.1080/14756366.2016.1238363. Epub 2016 Oct 21. J Enzyme Inhib Med Chem. 2017. PMID: 27766891 Free PMC article.

7

Pharmacophore Models and Pharmacophore-Based Virtual Screening: Concepts and Applications Exemplified on Hydroxysteroid Dehydrogenases.

Kaserer T, Beck KR, Akram M, Odermatt A, Schuster D. Kaserer T, et al. Molecules. 2015 Dec 19;20(12):22799-832. doi: 10.3390/molecules201219880. Molecules. 2015. PMID: 26703541 Free PMC article. Review.

8

Potential Antiosteoporotic Natural Product Lead Compounds That Inhibit 17β-Hydroxysteroid Dehydrogenase Type 2.

Vuorinen A, Engeli RT, Leugger S, Bachmann F, Akram M, Atanasov AG, Waltenberger B, Temml V, Stuppner H, Krenn L, Ateba SB, Njamen D, Davis RA, Odermatt A, Schuster D. Vuorinen A, et al. J Nat Prod. 2017 Apr 28;80(4):965-974. doi: 10.1021/acs.jnatprod.6b00950. Epub 2017 Mar 20. J Nat Prod. 2017. PMID: 28319389 Free PMC article.

9

A combinatorial approach for the discovery of cytochrome P450 2D6 inhibitors from nature.

Hochleitner J, Akram M, Ueberall M, Davis RA, Waltenberger B, Stuppner H, Sturm S, Ueberall F, Gostner JM, Schuster D. Hochleitner J, et al. Sci Rep. 2017 Aug 14;7(1):8071. doi: 10.1038/s41598-017-08404-0. Sci Rep. 2017. PMID: 28808272 Free PMC article.

10

Identification of the fungicide epoxiconazole by virtual screening and biological assessment as inhibitor of human 11β-hydroxylase and aldosterone synthase.

Akram M, Patt M, Kaserer T, Temml V, Waratchareeyakul W, Kratschmar DV, Haupenthal J, Hartmann RW, Odermatt A, Schuster D. Akram M, et al. J Steroid Biochem Mol Biol. 2019 Sep;192:105358. doi: 10.1016/j.jsbmb.2019.04.007. Epub 2019 Apr 6. J Steroid Biochem Mol Biol. 2019. PMID: 30965118

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