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Characterisation of UBP296: a novel, potent and selective kainate receptor antagonist.
More JC, Nistico R, Dolman NP, Clarke VR, Alt AJ, Ogden AM, Buelens FP, Troop HM, Kelland EE, Pilato F, Bleakman D, Bortolotto ZA, Collingridge GL, Jane DE. More JC, et al. Among authors: bleakman d. Neuropharmacology. 2004 Jul;47(1):46-64. doi: 10.1016/j.neuropharm.2004.03.005. Neuropharmacology. 2004. PMID: 15165833
Synthesis and pharmacological characterization of N3-substituted willardiine derivatives: role of the substituent at the 5-position of the uracil ring in the development of highly potent and selective GLUK5 kainate receptor antagonists.
Dolman NP, More JC, Alt A, Knauss JL, Pentikäinen OT, Glasser CR, Bleakman D, Mayer ML, Collingridge GL, Jane DE. Dolman NP, et al. Among authors: bleakman d. J Med Chem. 2007 Apr 5;50(7):1558-70. doi: 10.1021/jm061041u. Epub 2007 Mar 10. J Med Chem. 2007. PMID: 17348638
ACET is a highly potent and specific kainate receptor antagonist: characterisation and effects on hippocampal mossy fibre function.
Dargan SL, Clarke VR, Alushin GM, Sherwood JL, Nisticò R, Bortolotto ZA, Ogden AM, Bleakman D, Doherty AJ, Lodge D, Mayer ML, Fitzjohn SM, Jane DE, Collingridge GL. Dargan SL, et al. Among authors: bleakman d. Neuropharmacology. 2009 Jan;56(1):121-30. doi: 10.1016/j.neuropharm.2008.08.016. Epub 2008 Aug 22. Neuropharmacology. 2009. PMID: 18789344 Free PMC article.
Anxiolytic-like effects through a GLUK5 kainate receptor mechanism.
Alt A, Weiss B, Ornstein PL, Gleason SD, Bleakman D, Stratford RE Jr, Witkin JM. Alt A, et al. Among authors: bleakman d. Neuropharmacology. 2007 Jun;52(7):1482-7. doi: 10.1016/j.neuropharm.2007.02.005. Epub 2007 Mar 2. Neuropharmacology. 2007. PMID: 17418283
A hippocampal GluR5 kainate receptor regulating inhibitory synaptic transmission.
Clarke VR, Ballyk BA, Hoo KH, Mandelzys A, Pellizzari A, Bath CP, Thomas J, Sharpe EF, Davies CH, Ornstein PL, Schoepp DD, Kamboj RK, Collingridge GL, Lodge D, Bleakman D. Clarke VR, et al. Among authors: bleakman d. Nature. 1997 Oct 9;389(6651):599-603. doi: 10.1038/39315. Nature. 1997. PMID: 9335499
92 results