Ciesielski F - Search Results

1

Common architecture of nuclear receptor heterodimers on DNA direct repeat elements with different spacings.

Rochel N, Ciesielski F, Godet J, Moman E, Roessle M, Peluso-Iltis C, Moulin M, Haertlein M, Callow P, Mély Y, Svergun DI, Moras D. Rochel N, et al. Among authors: ciesielski f. Nat Struct Mol Biol. 2011 May;18(5):564-70. doi: 10.1038/nsmb.2054. Epub 2011 Apr 10. Nat Struct Mol Biol. 2011. PMID: 21478865

2

Structural investigation of the ligand binding domain of the zebrafish VDR in complexes with 1alpha,25(OH)2D3 and Gemini: purification, crystallization and preliminary X-ray diffraction analysis.

Ciesielski F, Rochel N, Mitschler A, Kouzmenko A, Moras D. Ciesielski F, et al. J Steroid Biochem Mol Biol. 2004 May;89-90(1-5):55-9. doi: 10.1016/j.jsbmb.2004.03.109. J Steroid Biochem Mol Biol. 2004. PMID: 15225747

3

Adaptability of the Vitamin D nuclear receptor to the synthetic ligand Gemini: remodelling the LBP with one side chain rotation.

Ciesielski F, Rochel N, Moras D. Ciesielski F, et al. J Steroid Biochem Mol Biol. 2007 Mar;103(3-5):235-42. doi: 10.1016/j.jsbmb.2006.12.003. Epub 2007 Jan 10. J Steroid Biochem Mol Biol. 2007. PMID: 17218092

4

Structure-based design of a superagonist ligand for the vitamin D nuclear receptor.

Hourai S, Rodrigues LC, Antony P, Reina-San-Martin B, Ciesielski F, Magnier BC, Schoonjans K, Mouriño A, Rochel N, Moras D. Hourai S, et al. Among authors: ciesielski f. Chem Biol. 2008 Apr;15(4):383-92. doi: 10.1016/j.chembiol.2008.03.016. Chem Biol. 2008. PMID: 18420145

5

Structural basis for the accommodation of bis- and tris-aromatic derivatives in vitamin D nuclear receptor.

Ciesielski F, Sato Y, Chebaro Y, Moras D, Dejaegere A, Rochel N. Ciesielski F, et al. J Med Chem. 2012 Oct 11;55(19):8440-9. doi: 10.1021/jm300858s. Epub 2012 Sep 19. J Med Chem. 2012. PMID: 22957834

6

A vitamin D receptor selectively activated by gemini analogs reveals ligand dependent and independent effects.

Huet T, Laverny G, Ciesielski F, Molnár F, Ramamoorthy TG, Belorusova AY, Antony P, Potier N, Metzger D, Moras D, Rochel N. Huet T, et al. Among authors: ciesielski f. Cell Rep. 2015 Feb 3;10(4):516-26. doi: 10.1016/j.celrep.2014.12.045. Epub 2015 Jan 22. Cell Rep. 2015. PMID: 25620699 Free article.

7

Structural basis of synthetic agonist activation of the nuclear receptor REV-ERB.

Murray MH, Valfort AC, Koelblen T, Ronin C, Ciesielski F, Chatterjee A, Veerakanellore GB, Elgendy B, Walker JK, Hegazy L, Burris TP. Murray MH, et al. Among authors: ciesielski f. Nat Commun. 2022 Nov 21;13(1):7131. doi: 10.1038/s41467-022-34892-4. Nat Commun. 2022. PMID: 36414641 Free PMC article.

8

Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists.

Ouvry G, Bouix-Peter C, Ciesielski F, Chantalat L, Christin O, Comino C, Duvert D, Feret C, Harris CS, Lamy L, Luzy AP, Musicki B, Orfila D, Pascau J, Parnet V, Perrin A, Pierre R, Polge G, Raffin C, Rival Y, Taquet N, Thoreau E, Hennequin LF. Ouvry G, et al. Among authors: ciesielski f. Bioorg Med Chem Lett. 2016 Dec 1;26(23):5802-5808. doi: 10.1016/j.bmcl.2016.10.023. Epub 2016 Oct 12. Bioorg Med Chem Lett. 2016. PMID: 27815118

9

Triazolopyridines as selective JAK1 inhibitors: from hit identification to GLPG0634.

Menet CJ, Fletcher SR, Van Lommen G, Geney R, Blanc J, Smits K, Jouannigot N, Deprez P, van der Aar EM, Clement-Lacroix P, Lepescheux L, Galien R, Vayssiere B, Nelles L, Christophe T, Brys R, Uhring M, Ciesielski F, Van Rompaey L. Menet CJ, et al. Among authors: ciesielski f. J Med Chem. 2014 Nov 26;57(22):9323-42. doi: 10.1021/jm501262q. Epub 2014 Nov 17. J Med Chem. 2014. PMID: 25369270

10

Biophysical and structural characterization of mono/di-arylated lactosamine derivatives interaction with human galectin-3.

Atmanene C, Ronin C, Téletchéa S, Gautier FM, Djedaïni-Pilard F, Ciesielski F, Vivat V, Grandjean C. Atmanene C, et al. Among authors: ciesielski f. Biochem Biophys Res Commun. 2017 Jul 29;489(3):281-286. doi: 10.1016/j.bbrc.2017.05.150. Epub 2017 May 26. Biochem Biophys Res Commun. 2017. PMID: 28554839

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