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Covalent targeting of remote cysteine residues to develop CDK12 and CDK13 inhibitors.
Nat Chem Biol. 2016 Oct;12(10):876-84. doi: 10.1038/nchembio.2166. Epub 2016 Aug 29.
Nat Chem Biol. 2016.
PMID: 27571479
Free PMC article.
Structure-activity relationship study of THZ531 derivatives enables the discovery of BSJ-01-175 as a dual CDK12/13 covalent inhibitor with efficacy in Ewing sarcoma.
Jiang B, Jiang J, Kaltheuner IH, Iniguez AB, Anand K, Ferguson FM, Ficarro SB, Seong BKA, Greifenberg AK, Dust S, Kwiatkowski NP, Marto JA, Stegmaier K, Zhang T, Geyer M, Gray NS.
Jiang B, et al. Among authors: greifenberg ak.
Eur J Med Chem. 2021 Oct 5;221:113481. doi: 10.1016/j.ejmech.2021.113481. Epub 2021 Apr 20.
Eur J Med Chem. 2021.
PMID: 33945934
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Structural and Functional Analysis of the Cdk13/Cyclin K Complex.
Greifenberg AK, Hönig D, Pilarova K, Düster R, Bartholomeeusen K, Bösken CA, Anand K, Blazek D, Geyer M.
Greifenberg AK, et al.
Cell Rep. 2016 Jan 12;14(2):320-31. doi: 10.1016/j.celrep.2015.12.025. Epub 2015 Dec 31.
Cell Rep. 2016.
PMID: 26748711
Free article.
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CDK12 Inhibition Reverses De Novo and Acquired PARP Inhibitor Resistance in BRCA Wild-Type and Mutated Models of Triple-Negative Breast Cancer.
Johnson SF, Cruz C, Greifenberg AK, Dust S, Stover DG, Chi D, Primack B, Cao S, Bernhardy AJ, Coulson R, Lazaro JB, Kochupurakkal B, Sun H, Unitt C, Moreau LA, Sarosiek KA, Scaltriti M, Juric D, Baselga J, Richardson AL, Rodig SJ, D'Andrea AD, Balmaña J, Johnson N, Geyer M, Serra V, Lim E, Shapiro GI.
Johnson SF, et al. Among authors: greifenberg ak.
Cell Rep. 2016 Nov 22;17(9):2367-2381. doi: 10.1016/j.celrep.2016.10.077.
Cell Rep. 2016.
PMID: 27880910
Free PMC article.
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P-TEFb regulation of transcription termination factor Xrn2 revealed by a chemical genetic screen for Cdk9 substrates.
Sansó M, Levin RS, Lipp JJ, Wang VY, Greifenberg AK, Quezada EM, Ali A, Ghosh A, Larochelle S, Rana TM, Geyer M, Tong L, Shokat KM, Fisher RP.
Sansó M, et al. Among authors: greifenberg ak.
Genes Dev. 2016 Jan 1;30(1):117-31. doi: 10.1101/gad.269589.115.
Genes Dev. 2016.
PMID: 26728557
Free PMC article.
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Brd4 activates P-TEFb for RNA polymerase II CTD phosphorylation.
Itzen F, Greifenberg AK, Bösken CA, Geyer M.
Itzen F, et al. Among authors: greifenberg ak.
Nucleic Acids Res. 2014 Jul;42(12):7577-90. doi: 10.1093/nar/gku449. Epub 2014 May 23.
Nucleic Acids Res. 2014.
PMID: 24860166
Free PMC article.
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Ubiquitin-Dependent Turnover of MYC Antagonizes MYC/PAF1C Complex Accumulation to Drive Transcriptional Elongation.
Jaenicke LA, von Eyss B, Carstensen A, Wolf E, Xu W, Greifenberg AK, Geyer M, Eilers M, Popov N.
Jaenicke LA, et al. Among authors: greifenberg ak.
Mol Cell. 2016 Jan 7;61(1):54-67. doi: 10.1016/j.molcel.2015.11.007. Epub 2015 Dec 10.
Mol Cell. 2016.
PMID: 26687678
Free article.
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MIR sequences recruit zinc finger protein ZNF768 to expressed genes.
Rohrmoser M, Kluge M, Yahia Y, Gruber-Eber A, Maqbool MA, Forné I, Krebs S, Blum H, Greifenberg AK, Geyer M, Descostes N, Imhof A, Andrau JC, Friedel CC, Eick D.
Rohrmoser M, et al. Among authors: greifenberg ak.
Nucleic Acids Res. 2019 Jan 25;47(2):700-715. doi: 10.1093/nar/gky1148.
Nucleic Acids Res. 2019.
PMID: 30476274
Free PMC article.
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