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Extended structure-activity relationship and pharmacokinetic investigation of (4-quinolinoyl)glycyl-2-cyanopyrrolidine inhibitors of fibroblast activation protein (FAP).
J Med Chem. 2014 Apr 10;57(7):3053-74. doi: 10.1021/jm500031w. Epub 2014 Mar 24.
J Med Chem. 2014.
PMID: 24617858
Selective Inhibitors of Fibroblast Activation Protein (FAP) with a (4-Quinolinoyl)-glycyl-2-cyanopyrrolidine Scaffold.
Jansen K, Heirbaut L, Cheng JD, Joossens J, Ryabtsova O, Cos P, Maes L, Lambeir AM, De Meester I, Augustyns K, Van der Veken P.
Jansen K, et al. Among authors: heirbaut l.
ACS Med Chem Lett. 2013 Mar 18;4(5):491-6. doi: 10.1021/ml300410d. eCollection 2013 May 9.
ACS Med Chem Lett. 2013.
PMID: 24900696
Free PMC article.
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