Inagaki H - Search Results

1

Design, Synthesis, and Biological Evaluation of Novel 7-[(3 aS,7 aS)-3 a-Aminohexahydropyrano[3,4- c]pyrrol-2(3 H)-yl]-8-methoxyquinolines with Potent Antibacterial Activity against Respiratory Pathogens.

Odagiri T, Inagaki H, Nagamochi M, Kitamura T, Komoriya S, Takahashi H. Odagiri T, et al. Among authors: inagaki h. J Med Chem. 2018 Aug 23;61(16):7234-7244. doi: 10.1021/acs.jmedchem.8b00644. Epub 2018 Aug 8. J Med Chem. 2018. PMID: 30063826

2

Synthesis and structure-activity relationships of 5-amino-6-fluoro-1-[(1R,2S)-2-fluorocyclopropan-1-yl]-8-methylquinolonecarboxylic acid antibacterials having fluorinated 7-[(3R)-3-(1-aminocyclopropan-1-yl)pyrrolidin-1-yl] substituents.

Inagaki H, Miyauchi S, Miyauchi RN, Kawato HC, Ohki H, Matsuhashi N, Kawakami K, Takahashi H, Takemura M. Inagaki H, et al. J Med Chem. 2003 Mar 13;46(6):1005-15. doi: 10.1021/jm020328y. J Med Chem. 2003. PMID: 12620077

3

Synthesis and antibacterial activity of novel 6-fluoro-1-[(1R,2S)-2-fluorocyclopropan-1-yl]-4-oxoquinoline-3-carboxylic acids bearing cyclopropane-fused 2-amino-8-azabicyclo[4.3.0]nonan-8-yl substituents at the C-7 position.

Inagaki H, Takahashi H, Takemura M. Inagaki H, et al. Bioorg Med Chem Lett. 2004 Oct 18;14(20):5193-8. doi: 10.1016/j.bmcl.2004.07.064. Bioorg Med Chem Lett. 2004. PMID: 15380226

4

Design, synthesis and biological evaluations of novel 7-[3-(1-aminocycloalkyl)pyrrolidin-1-yl]-6-desfluoro-8-methoxyquinolones with potent antibacterial activity against multi-drug resistant Gram-positive bacteria.

Miyauchi R, Kawakami K, Ito M, Matsuhashi N, Ohki H, Inagaki H, Takahashi H, Takemura M. Miyauchi R, et al. Among authors: inagaki h. Bioorg Med Chem. 2009 Oct 1;17(19):6879-89. doi: 10.1016/j.bmc.2009.08.026. Epub 2009 Aug 20. Bioorg Med Chem. 2009. PMID: 19736016

5

Design, synthesis, and biological evaluations of novel 7-[7-amino-7-methyl-5-azaspiro[2.4]heptan-5-yl]-8-methoxyquinolines with potent antibacterial activity against respiratory pathogens.

Odagiri T, Inagaki H, Sugimoto Y, Nagamochi M, Miyauchi RN, Kuroyanagi J, Kitamura T, Komoriya S, Takahashi H. Odagiri T, et al. Among authors: inagaki h. J Med Chem. 2013 Mar 14;56(5):1974-83. doi: 10.1021/jm301650g. Epub 2013 Feb 25. J Med Chem. 2013. PMID: 23409972

6

Discovery of Novel 7-[(1R,5S)-1-Amino-5-fluoro-3-azabicyclo[3.3.0]octan-3-yl]-6-fluoro-1-[(1R,2S)-2-fluorocyclopropane]-8-(methoxy or methyl)quinolones.

Komoriya S, Odagiri T, Inagaki H, Nagamochi M, Miyauchi R, Yoshida KI, Kitamura T, Takahashi H. Komoriya S, et al. Among authors: inagaki h. Chem Pharm Bull (Tokyo). 2019;67(1):47-58. doi: 10.1248/cpb.c18-00671. Chem Pharm Bull (Tokyo). 2019. PMID: 30606950 Free article.

7

Discovery of Novel Pyrido-pyridazinone Derivatives as FER Tyrosine Kinase Inhibitors with Antitumor Activity.

Taniguchi T, Inagaki H, Baba D, Yasumatsu I, Toyota A, Kaneta Y, Kiga M, Iimura S, Odagiri T, Shibata Y, Ueda K, Seo M, Shimizu H, Imaoka T, Nakayama K. Taniguchi T, et al. Among authors: inagaki h. ACS Med Chem Lett. 2019 Mar 15;10(5):737-742. doi: 10.1021/acsmedchemlett.8b00631. eCollection 2019 May 9. ACS Med Chem Lett. 2019. PMID: 31097992 Free PMC article.

8

Synthesis and antifungal activity of rhodopeptin analogues. 2. Modification of the west amino acid moiety.

Nakayama K, Kawato HC, Inagaki H, Nakajima R, Kitamura A, Someya K, Ohta T. Nakayama K, et al. Among authors: inagaki h. Org Lett. 2000 Apr 6;2(7):977-80. doi: 10.1021/ol005630k. Org Lett. 2000. PMID: 10768201

9

Novel peptidomimetics of the antifungal cyclic peptide Rhodopeptin: design of mimetics utilizing scaffolding methodology.

Nakayama K, Kawato HC, Inagaki H, Ohta T. Nakayama K, et al. Among authors: inagaki h. Org Lett. 2001 Nov 1;3(22):3447-50. doi: 10.1021/ol0163934. Org Lett. 2001. PMID: 11678679

10

Synthesis and antifungal activity of rhodopeptin analogues. 1. Modification of the east and south amino acid moieties.

Kawato HC, Nakayama K, Inagaki H, Nakajima R, Kitamura A, Someya K, Ohta T. Kawato HC, et al. Among authors: inagaki h. Org Lett. 2000 Apr 6;2(7):973-6. doi: 10.1021/ol005631c. Org Lett. 2000. PMID: 10768200

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