Jayaram HN - Search Results

1

Synthesis, conformational analysis, and biological activity of new analogues of thiazole-4-carboxamide adenine dinucleotide (TAD) as IMP dehydrogenase inhibitors.

Franchetti P, Cappellacci L, Pasqualini M, Petrelli R, Jayaprakasan V, Jayaram HN, Boyd DB, Jain MD, Grifantini M. Franchetti P, et al. Among authors: jayaram hn. Bioorg Med Chem. 2005 Mar 15;13(6):2045-53. doi: 10.1016/j.bmc.2005.01.007. Bioorg Med Chem. 2005. PMID: 15727858

2

Antitumor activity of C-methyl-beta-D-ribofuranosyladenine nucleoside ribonucleotide reductase inhibitors.

Franchetti P, Cappellacci L, Pasqualini M, Petrelli R, Vita P, Jayaram HN, Horvath Z, Szekeres T, Grifantini M. Franchetti P, et al. Among authors: jayaram hn. J Med Chem. 2005 Jul 28;48(15):4983-9. doi: 10.1021/jm048944c. J Med Chem. 2005. PMID: 16033277

3

Ribose-modified purine nucleosides as ribonucleotide reductase inhibitors. Synthesis, antitumor activity, and molecular modeling of N6-substituted 3'-C-methyladenosine derivatives.

Cappellacci L, Franchetti P, Vita P, Petrelli R, Lavecchia A, Jayaram HN, Saiko P, Graser G, Szekeres T, Grifantini M. Cappellacci L, et al. Among authors: jayaram hn. J Med Chem. 2008 Jul 24;51(14):4260-9. doi: 10.1021/jm800205c. Epub 2008 Jun 28. J Med Chem. 2008. PMID: 18588281

4

Synthesis and biological activity of novel N6-substituted and 2,N6-disubstituted adenine ribo- and 3'-C-methyl-ribonucleosides as antitumor agents.

Cappellacci L, Petrelli R, Franchetti P, Vita P, Kusumanchi P, Kumar M, Jayaram HN, Zhou B, Yen Y, Grifantini M. Cappellacci L, et al. Among authors: jayaram hn. Eur J Med Chem. 2011 May;46(5):1499-504. doi: 10.1016/j.ejmech.2011.01.055. Epub 2011 Feb 3. Eur J Med Chem. 2011. PMID: 21349610

5

From the covalent linkage of drugs to novel inhibitors of ribonucleotide reductase: synthesis and biological evaluation of valproic esters of 3'-C-methyladenosine.

Petrelli R, Meli M, Vita P, Torquati I, Ferro A, Vodnala M, D'Alessandro N, Tolomeo M, Del Bello F, Kusumanchi P, Franchetti P, Grifantini M, Jayaram HN, Hofer A, Cappellacci L. Petrelli R, et al. Among authors: jayaram hn. Bioorg Med Chem Lett. 2014 Nov 15;24(22):5304-9. doi: 10.1016/j.bmcl.2014.09.046. Epub 2014 Sep 28. Bioorg Med Chem Lett. 2014. PMID: 25304896

6

Furanfurin and thiophenfurin: two novel tiazofurin analogues. Synthesis, structure, antitumor activity, and interactions with inosine monophosphate dehydrogenase.

Franchetti P, Cappellacci L, Grifantini M, Barzi A, Nocentini G, Yang H, O'Connor A, Jayaram HN, Carrell C, Goldstein BM. Franchetti P, et al. Among authors: jayaram hn. J Med Chem. 1995 Sep 15;38(19):3829-37. doi: 10.1021/jm00019a013. J Med Chem. 1995. PMID: 7562914

7

Synthesis, structure, and antiproliferative activity of selenophenfurin, an inosine 5'-monophosphate dehydrogenase inhibitor analogue of selenazofurin.

Franchetti P, Cappellacci L, Sheikha GA, Jayaram HN, Gurudutt VV, Sint T, Schneider BP, Jones WD, Goldstein BM, Perra G, De Montis A, Loi AG, La Colla P, Grifantini M. Franchetti P, et al. Among authors: jayaram hn. J Med Chem. 1997 May 23;40(11):1731-7. doi: 10.1021/jm960864o. J Med Chem. 1997. PMID: 9171883

8

Isosteric analogues of nicotinamide adenine dinucleotide derived from furanfurin, thiophenfurin, and selenophenfurin as mammalian inosine monophosphate dehydrogenase (type I and II) inhibitors.

Franchetti P, Cappellacci L, Perlini P, Jayaram HN, Butler A, Schneider BP, Collart FR, Huberman E, Grifantini M. Franchetti P, et al. Among authors: jayaram hn. J Med Chem. 1998 May 7;41(10):1702-7. doi: 10.1021/jm970772e. J Med Chem. 1998. PMID: 9572896

9

Synthesis, conformational analysis, and biological activity of C-thioribonucleosides related to tiazofurin.

Franchetti P, Marchetti S, Cappellacci L, Jayaram HN, Yalowitz JA, Goldstein BM, Barascut JL, Dukhan D, Imbach JL, Grifantini M. Franchetti P, et al. Among authors: jayaram hn. J Med Chem. 2000 Apr 6;43(7):1264-70. doi: 10.1021/jm990257b. J Med Chem. 2000. PMID: 10753464

10

A new C-nucleoside analogue of tiazofurin: synthesis and biological evaluation of 2-beta-D-ribofuranosylimidazole-4-carboxamide (imidazofurin).

Franchetti P, Marchetti S, Cappellacci L, Yalowitz JA, Jayaram HN, Goldstein BM, Grifantini M. Franchetti P, et al. Among authors: jayaram hn. Bioorg Med Chem Lett. 2001 Jan 8;11(1):67-9. doi: 10.1016/s0960-894x(00)00594-1. Bioorg Med Chem Lett. 2001. PMID: 11140736

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