Michejda CJ - Search Results

1

Design and synthesis of novel and potent inhibitors of the type II transmembrane serine protease, matriptase, based upon the sunflower trypsin inhibitor-1.

Li P, Jiang S, Lee SL, Lin CY, Johnson MD, Dickson RB, Michejda CJ, Roller PP. Li P, et al. Among authors: michejda cj. J Med Chem. 2007 Nov 29;50(24):5976-83. doi: 10.1021/jm0704898. Epub 2007 Nov 7. J Med Chem. 2007. PMID: 17985858

2

Design and synthesis of paclitaxel conjugated with an ErbB2-recognizing peptide, EC-1.

Li P, Jiang S, Pero SC, Oligino L, Krag DN, Michejda CJ, Roller PP. Li P, et al. Among authors: michejda cj. Biopolymers. 2007 Nov;87(4):225-30. doi: 10.1002/bip.20828. Biopolymers. 2007. PMID: 17879382

3

Rationally designed inhibitors identify STAT3 N-domain as a promising anticancer drug target.

Timofeeva OA, Gaponenko V, Lockett SJ, Tarasov SG, Jiang S, Michejda CJ, Perantoni AO, Tarasova NI. Timofeeva OA, et al. Among authors: michejda cj. ACS Chem Biol. 2007 Dec 21;2(12):799-809. doi: 10.1021/cb700186x. ACS Chem Biol. 2007. PMID: 18154267

4

Synthesis, biological activity, and crystal structure of potent nonnucleoside inhibitors of HIV-1 reverse transcriptase that retain activity against mutant forms of the enzyme.

Morningstar ML, Roth T, Farnsworth DW, Smith MK, Watson K, Buckheit RW Jr, Das K, Zhang W, Arnold E, Julias JG, Hughes SH, Michejda CJ. Morningstar ML, et al. Among authors: michejda cj. J Med Chem. 2007 Aug 23;50(17):4003-15. doi: 10.1021/jm060103d. Epub 2007 Jul 31. J Med Chem. 2007. PMID: 17663538 Free PMC article.

5

Transmembrane inhibitors of P-glycoprotein, an ABC transporter.

Tarasova NI, Seth R, Tarasov SG, Kosakowska-Cholody T, Hrycyna CA, Gottesman MM, Michejda CJ. Tarasova NI, et al. Among authors: michejda cj. J Med Chem. 2005 Jun 2;48(11):3768-75. doi: 10.1021/jm049065t. J Med Chem. 2005. PMID: 15916428

6

Stereoselectivity in the microsomal conversion of N-nitrosodimethylamine to formaldehyde.

Keefer LK, Kroeger-Koepke MB, Ishizaki H, Michejda CJ, Saavedra JE, Hrabie JA, Yang CS, Roller PP. Keefer LK, et al. Among authors: michejda cj. Chem Res Toxicol. 1990 Nov-Dec;3(6):540-4. doi: 10.1021/tx00018a008. Chem Res Toxicol. 1990. PMID: 2103325

7

Optimization of naphthalimide-imidazoacridone with potent antitumor activity leading to clinical candidate (HKH40A, RTA 502).

Hariprakasha HK, Kosakowska-Cholody T, Meyer C, Cholody WM, Stinson SF, Tarasova NI, Michejda CJ. Hariprakasha HK, et al. Among authors: michejda cj. J Med Chem. 2007 Nov 15;50(23):5557-60. doi: 10.1021/jm7009777. Epub 2007 Oct 16. J Med Chem. 2007. PMID: 17939651

8

Synthesis and biological activity of novel nonnucleoside inhibitors of HIV-1 reverse transcriptase. 2-Aryl-substituted benzimidazoles.

Roth T, Morningstar ML, Boyer PL, Hughes SH, Buckheit RW Jr, Michejda CJ. Roth T, et al. Among authors: michejda cj. J Med Chem. 1997 Dec 19;40(26):4199-207. doi: 10.1021/jm970096g. J Med Chem. 1997. PMID: 9435891

9

Molecular modeling calculations of HIV-1 reverse transcriptase nonnucleoside inhibitors: correlation of binding energy with biological activity for novel 2-aryl-substituted benzimidazole analogues.

Kroeger Smith MB, Hose BM, Hawkins A, Lipchock J, Farnsworth DW, Rizzo RC, Tirado-Rives J, Arnold E, Zhang W, Hughes SH, Jorgensen WL, Michejda CJ, Smith RH Jr. Kroeger Smith MB, et al. Among authors: michejda cj. J Med Chem. 2003 May 8;46(10):1940-7. doi: 10.1021/jm020271f. J Med Chem. 2003. PMID: 12723956

10

Structure-activity relationship studies for the peptide portion of the bladder epithelial cell antiproliferative factor from interstitial cystitis patients.

Kaczmarek P, Keay SK, Tocci GM, Koch KR, Zhang CO, Barchi JJ Jr, Grkovic D, Guo L, Michejda CJ. Kaczmarek P, et al. Among authors: michejda cj. J Med Chem. 2008 Oct 9;51(19):5974-83. doi: 10.1021/jm8002763. Epub 2008 Sep 13. J Med Chem. 2008. PMID: 18788730 Free PMC article.

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

86 results

Search Page