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Pyrrole-3-carboxamides as potent and selective JAK2 inhibitors.
Bioorg Med Chem. 2014 Sep 1;22(17):4998-5012. doi: 10.1016/j.bmc.2014.06.025. Epub 2014 Jun 21.
Bioorg Med Chem. 2014.
PMID: 25009002
Rational design, synthesis and characterization of potent, non-peptidic Smac mimics/XIAP inhibitors as proapoptotic agents for cancer therapy.
Seneci P, Bianchi A, Battaglia C, Belvisi L, Bolognesi M, Caprini A, Cossu F, Franco Ed, Matteo Md, Delia D, Drago C, Khaled A, Lecis D, Manzoni L, Marizzoni M, Mastrangelo E, Milani M, Motto I, Moroni E, Potenza D, Rizzo V, Servida F, Turlizzi E, Varrone M, Vasile F, Scolastico C.
Seneci P, et al. Among authors: motto i.
Bioorg Med Chem. 2009 Aug 15;17(16):5834-56. doi: 10.1016/j.bmc.2009.07.009. Epub 2009 Jul 10.
Bioorg Med Chem. 2009.
PMID: 19620011
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Discovery of 2-(cyclohexylmethylamino)pyrimidines as a new class of reversible valosine containing protein inhibitors.
Cervi G, Magnaghi P, Asa D, Avanzi N, Badari A, Borghi D, Caruso M, Cirla A, Cozzi L, Felder E, Galvani A, Gasparri F, Lomolino A, Magnuson S, Malgesini B, Motto I, Pasi M, Rizzi S, Salom B, Sorrentino G, Troiani S, Valsasina B, O'Brien T, Isacchi A, Donati D, D'Alessio R.
Cervi G, et al. Among authors: motto i.
J Med Chem. 2014 Dec 26;57(24):10443-54. doi: 10.1021/jm501313x. Epub 2014 Dec 12.
J Med Chem. 2014.
PMID: 25474526
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Novel pyrrole carboxamide inhibitors of JAK2 as potential treatment of myeloproliferative disorders.
Brasca MG, Gnocchi P, Nesi M, Amboldi N, Avanzi N, Bertrand J, Bindi S, Canevari G, Casero D, Ciomei M, Colombo N, Cribioli S, Fachin G, Felder ER, Galvani A, Isacchi A, Motto I, Panzeri A, Donati D.
Brasca MG, et al. Among authors: motto i.
Bioorg Med Chem. 2015 May 15;23(10):2387-407. doi: 10.1016/j.bmc.2015.03.059. Epub 2015 Mar 28.
Bioorg Med Chem. 2015.
PMID: 25882525
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Discovery and optimization of 4-pyrazolyl-2-aminopyrimidine derivatives as potent spleen tyrosine kinase (SYK) inhibitors.
Cervi G, D'Alessio R, Bindi S, Buffa L, Burocchi A, Canevari G, Modugno M, Motto I, Saturno G, Orsini P.
Cervi G, et al. Among authors: motto i.
Eur J Med Chem. 2024 Apr 15;270:116375. doi: 10.1016/j.ejmech.2024.116375. Epub 2024 Apr 4.
Eur J Med Chem. 2024.
PMID: 38604095
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Molecular Dynamics Simulations of p97 Including Covalent, Allosteric and ATP-competitive Inhibitors.
Rendine S, Orrenius C, Dapiaggi F, Pieraccini S, Motto I, D'Alessio R, Magnaghi P, Isacchi A, Felder E, Sironi M.
Rendine S, et al. Among authors: motto i.
Acta Chim Slov. 2019 Jun;66(2):395-401.
Acta Chim Slov. 2019.
PMID: 33855508
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Grafting aminocyclopentane carboxylic acids onto the RGD tripeptide sequence generates low nanomolar alphaVbeta3/alphaVbeta5 integrin dual binders.
Casiraghi G, Rassu G, Auzzas L, Burreddu P, Gaetani E, Battistini L, Zanardi F, Curti C, Nicastro G, Belvisi L, Motto I, Castorina M, Giannini G, Pisano C.
Casiraghi G, et al. Among authors: motto i.
J Med Chem. 2005 Dec 1;48(24):7675-87. doi: 10.1021/jm050698x.
J Med Chem. 2005.
PMID: 16302808
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New aryl hydrocarbon receptor homology model targeted to improve docking reliability.
Motto I, Bordogna A, Soshilov AA, Denison MS, Bonati L.
Motto I, et al.
J Chem Inf Model. 2011 Nov 28;51(11):2868-81. doi: 10.1021/ci2001617. Epub 2011 Nov 2.
J Chem Inf Model. 2011.
PMID: 21981577
Free PMC article.
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