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From Combinations to Single-Molecule Polypharmacology-Cromolyn-Ibuprofen Conjugates for Alzheimer's Disease.
Molecules. 2021 Feb 19;26(4):1112. doi: 10.3390/molecules26041112.
Molecules. 2021.
PMID: 33669839
Free PMC article.
Taking inspiration from an ongoing clinical trial, this work aims to convert a promising cromolyn-ibuprofen drug combination into single-molecule "codrugs." Such codrugs should be able to similarly modulate neuroinflammatory and amyloid pathways, while showing peculiar pro …
Taking inspiration from an ongoing clinical trial, this work aims to convert a promising cromolyn-ibuprofen drug combination into single- …
New Coumarin Derivatives as Cholinergic and Cannabinoid System Modulators.
Montanari S, Allarà M, Scalvini L, Kostrzewa M, Belluti F, Gobbi S, Naldi M, Rivara S, Bartolini M, Ligresti A, Bisi A, Rampa A.
Montanari S, et al.
Molecules. 2021 May 28;26(11):3254. doi: 10.3390/molecules26113254.
Molecules. 2021.
PMID: 34071439
Free PMC article.
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Bio-Guided Fractionation of Stem Bark Extracts from Phyllanthus muellarianus: Identification of Phytocomponents with Anti-Cholinesterase Activity.
Naldi M, Brusotti G, Massolini G, Andrisano V, Temporini C, Bartolini M.
Naldi M, et al.
Molecules. 2021 Jul 20;26(14):4376. doi: 10.3390/molecules26144376.
Molecules. 2021.
PMID: 34299650
Free PMC article.
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