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Design and Characterization of 1,3-Dihydro-2H-benzo[d]azepin-2-ones as Rule-of-5 Compliant Bivalent BET Inhibitors.
ACS Med Chem Lett. 2023 Aug 14;14(9):1231-1236. doi: 10.1021/acsmedchemlett.3c00242. eCollection 2023 Sep 14.
ACS Med Chem Lett. 2023.
PMID: 37736196
Exploitation of a Novel Binding Pocket in Human Lipoprotein-Associated Phospholipase A2 (Lp-PLA2) Discovered through X-ray Fragment Screening.
Woolford AJ, Pero JE, Aravapalli S, Berdini V, Coyle JE, Day PJ, Dodson AM, Grondin P, Holding FP, Lee LY, Li P, Manas ES, Marino J Jr, Martin AC, McCleland BW, McMenamin RL, Murray CW, Neipp CE, Page LW, Patel VK, Potvain F, Rich S, Rivero RA, Smith K, Somers DO, Trottet L, Velagaleti R, Williams G, Xie R.
Woolford AJ, et al. Among authors: neipp ce.
J Med Chem. 2016 Jun 9;59(11):5356-67. doi: 10.1021/acs.jmedchem.6b00212. Epub 2016 May 20.
J Med Chem. 2016.
PMID: 27167608
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Synthesis of bridged azabicyclic structures via ring-closing olefin metathesis.
Neipp CE, Martin SF.
Neipp CE, et al.
J Org Chem. 2003 Nov 14;68(23):8867-78. doi: 10.1021/jo0349936.
J Org Chem. 2003.
PMID: 14604356
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The synthesis of homoallylic amines utilizing a cuprate-based 1,2-metalate rearrangement.
Neipp CE, Humphrey JM, Martin SF.
Neipp CE, et al.
J Org Chem. 2001 Jan 26;66(2):531-7. doi: 10.1021/jo001386z.
J Org Chem. 2001.
PMID: 11429825
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