Pockes S - Search Results

1

Development of a Conformational Histamine H₃ Receptor Biosensor for the Synchronous Screening of Agonists and Inverse Agonists.

Schihada H, Ma X, Zabel U, Vischer HF, Schulte G, Leurs R, Pockes S, Lohse MJ. Schihada H, et al. Among authors: pockes s. ACS Sens. 2020 Jun 26;5(6):1734-1742. doi: 10.1021/acssensors.0c00397. Epub 2020 May 28. ACS Sens. 2020. PMID: 32397705 Free PMC article.

2

Highly Potent, Stable, and Selective Dimeric Hetarylpropylguanidine-Type Histamine H₂ Receptor Agonists.

Pockes S, Wifling D, Keller M, Buschauer A, Elz S. Pockes S, et al. ACS Omega. 2018 Mar 31;3(3):2865-2882. doi: 10.1021/acsomega.8b00128. Epub 2018 Mar 9. ACS Omega. 2018. PMID: 30221224 Free PMC article.

3

Discovery of a G Protein-Biased Radioligand for the Histamine H₂ Receptor with Reversible Binding Properties.

Tropmann K, Höring C, Plank N, Pockes S. Tropmann K, et al. Among authors: pockes s. J Med Chem. 2020 Nov 12;63(21):13090-13102. doi: 10.1021/acs.jmedchem.0c01494. Epub 2020 Oct 27. J Med Chem. 2020. PMID: 33108724

4

A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes.

Höring C, Seibel U, Tropmann K, Grätz L, Mönnich D, Pitzl S, Bernhardt G, Pockes S, Strasser A. Höring C, et al. Among authors: pockes s. Int J Mol Sci. 2020 Nov 10;21(22):8440. doi: 10.3390/ijms21228440. Int J Mol Sci. 2020. PMID: 33182741 Free PMC article.

5

Structural modifications in the distal, regulatory region of histamine H₃ receptor antagonists leading to the identification of a potent anti-obesity agent.

Szczepańska K, Pockes S, Podlewska S, Höring C, Mika K, Latacz G, Bednarski M, Siwek A, Karcz T, Nagl M, Bresinsky M, Mönnich D, Seibel U, Kuder KJ, Kotańska M, Stark H, Elz S, Kieć-Kononowicz K. Szczepańska K, et al. Among authors: pockes s. Eur J Med Chem. 2021 Mar 5;213:113041. doi: 10.1016/j.ejmech.2020.113041. Epub 2020 Nov 24. Eur J Med Chem. 2021. PMID: 33261900

6

Histamine H₂ receptor radioligands: triumphs and challenges.

Pockes S, Tropmann K. Pockes S, et al. Future Med Chem. 2021 Jun;13(12):1073-1081. doi: 10.4155/fmc-2021-0058. Epub 2021 Apr 28. Future Med Chem. 2021. PMID: 33906421 Free article. Review.

7

A Versatile Sub-Nanomolar Fluorescent Ligand Enables NanoBRET Binding Studies and Single-Molecule Microscopy at the Histamine H₃ Receptor.

Rosier N, Grätz L, Schihada H, Möller J, Işbilir A, Humphrys LJ, Nagl M, Seibel U, Lohse MJ, Pockes S. Rosier N, et al. Among authors: pockes s. J Med Chem. 2021 Aug 12;64(15):11695-11708. doi: 10.1021/acs.jmedchem.1c01089. Epub 2021 Jul 26. J Med Chem. 2021. PMID: 34309390

8

Structural and Molecular Insight into Piperazine and Piperidine Derivatives as Histamine H₃ and Sigma-1 Receptor Antagonists with Promising Antinociceptive Properties.

Szczepańska K, Podlewska S, Dichiara M, Gentile D, Patamia V, Rosier N, Mönnich D, Ruiz Cantero MC, Karcz T, Łażewska D, Siwek A, Pockes S, Cobos EJ, Marrazzo A, Stark H, Rescifina A, Bojarski AJ, Amata E, Kieć-Kononowicz K. Szczepańska K, et al. Among authors: pockes s. ACS Chem Neurosci. 2022 Jan 5;13(1):1-15. doi: 10.1021/acschemneuro.1c00435. Epub 2021 Dec 15. ACS Chem Neurosci. 2022. PMID: 34908391 Free PMC article.

9

Development of Fluorescent AF64394 Analogues Enables Real-Time Binding Studies for the Orphan Class A GPCR GPR3.

Bresinsky M, Shahraki A, Kolb P, Pockes S, Schihada H. Bresinsky M, et al. Among authors: pockes s. J Med Chem. 2023 Nov 9;66(21):15025-15041. doi: 10.1021/acs.jmedchem.3c01707. Epub 2023 Oct 31. J Med Chem. 2023. PMID: 37907069 Free PMC article.

10

Fluorescent Tools for the Imaging of Dopamine D₂ -Like Receptors.

Nagl M, Mönnich D, Rosier N, Schihada H, Sirbu A, Konar N, Reyes-Resina I, Navarro G, Franco R, Kolb P, Annibale P, Pockes S. Nagl M, et al. Among authors: pockes s. Chembiochem. 2024 Jan 15;25(2):e202300659. doi: 10.1002/cbic.202300659. Epub 2023 Nov 20. Chembiochem. 2024. PMID: 37942961

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