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Effects of positional and geometrical isomerism on the biological activity of some novel oxazolidinones.
Bioorg Med Chem Lett. 2005 Jan 17;15(2):337-43. doi: 10.1016/j.bmcl.2004.10.073.
Bioorg Med Chem Lett. 2005.
PMID: 15603950
Substituent activity relationship studies on new azolo benzoxazepinyl oxazolidinones.
Das J, Sitaram Kumar M, Subrahmanyam D, Sastry TV, Prasad Narasimhulu C, Laxman Rao CV, Kannan M, Roshaiah M, Awasthi R, Patil SN, Sarnaik HM, Rao Mamidi NV, Selvakumar N, Iqbal J.
Das J, et al. Among authors: roshaiah m.
Bioorg Med Chem. 2006 Dec 1;14(23):8032-42. doi: 10.1016/j.bmc.2006.07.040. Epub 2006 Aug 10.
Bioorg Med Chem. 2006.
PMID: 16904333
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Discovery of novel, orally available benzimidazoles as melanin concentrating hormone receptor 1 (MCHR1) antagonists.
Sasmal PK, Sasmal S, Rao PT, Venkatesham B, Roshaiah M, Abbineni C, Khanna I, Jadhav VP, Suresh J, Talwar R, Muzeeb S, Receveur JM, Frimurer TM, Rist Ø, Elster L, Högberg T.
Sasmal PK, et al. Among authors: roshaiah m.
Bioorg Med Chem Lett. 2010 Sep 15;20(18):5443-8. doi: 10.1016/j.bmcl.2010.07.086. Epub 2010 Jul 29.
Bioorg Med Chem Lett. 2010.
PMID: 20724156
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Optimisation of in silico derived 2-aminobenzimidazole hits as unprecedented selective kappa opioid receptor agonists.
Sasmal PK, Krishna CV, Adabala SS, Roshaiah M, Rawoof KA, Thadi E, Sukumar KP, Cheera S, Abbineni C, Rao KV, Prasanthi A, Nijhawan K, Jaleel M, Iyer LR, Chaitanya TK, Tiwari NK, Krishna NL, Potluri V, Khanna I, Frimurer TM, Lückmann M, Rist Ø, Elster L, Högberg T.
Sasmal PK, et al. Among authors: roshaiah m.
Bioorg Med Chem Lett. 2015 Feb 15;25(4):887-92. doi: 10.1016/j.bmcl.2014.12.064. Epub 2015 Jan 6.
Bioorg Med Chem Lett. 2015.
PMID: 25599839
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