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Discovery of a series of potent arylthiadiazole H(3) antagonists.
Bioorg Med Chem Lett. 2011 Jan 15;21(2):861-4. doi: 10.1016/j.bmcl.2010.11.065. Epub 2010 Nov 21.
Bioorg Med Chem Lett. 2011.
PMID: 21186123
Fused bicycles as arylketone bioisosteres leading to potent, orally active thiadiazole H3 antagonists.
Xiao D, Palani A, Sofolarides M, Aslanian R, West RE Jr, Williams SM, Wu RL, Hwa J, Sondey C, Lachowicz J, Korfmacher WA.
Xiao D, et al. Among authors: sofolarides m.
Bioorg Med Chem Lett. 2012 May 1;22(9):3354-7. doi: 10.1016/j.bmcl.2012.02.076. Epub 2012 Mar 8.
Bioorg Med Chem Lett. 2012.
PMID: 22464130
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Conformation constraint of anilides enabling the discovery of tricyclic lactams as potent MK2 non-ATP competitive inhibitors.
Xiao D, Palani A, Huang X, Sofolarides M, Zhou W, Chen X, Aslanian R, Guo Z, Fossetta J, Tian F, Trivedi P, Spacciapoli P, Whitehurst CE, Lundell D.
Xiao D, et al. Among authors: sofolarides m.
Bioorg Med Chem Lett. 2013 Jun 1;23(11):3262-6. doi: 10.1016/j.bmcl.2013.03.109. Epub 2013 Apr 4.
Bioorg Med Chem Lett. 2013.
PMID: 23602398
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Discovery of SCH 900271, a Potent Nicotinic Acid Receptor Agonist for the Treatment of Dyslipidemia.
Palani A, Rao AU, Chen X, Huang X, Su J, Tang H, Huang Y, Qin J, Xiao D, Degrado S, Sofolarides M, Zhu X, Liu Z, McKittrick B, Zhou W, Aslanian R, Greenlee WJ, Senior M, Cheewatrakoolpong B, Zhang H, Farley C, Cook J, Kurowski S, Li Q, van Heek M, Wang G, Hsieh Y, Li F, Greenfeder S, Chintala M.
Palani A, et al. Among authors: sofolarides m.
ACS Med Chem Lett. 2011 Nov 24;3(1):63-8. doi: 10.1021/ml200243g. eCollection 2012 Jan 12.
ACS Med Chem Lett. 2011.
PMID: 24900372
Free PMC article.
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Discovery of a novel series of potent MK2 non-ATP competitive inhibitors using 1,2-substituted azoles as cis-amide isosteres.
Xiao D, Zhu X, Sofolarides M, Degrado S, Shao N, Rao A, Chen X, Aslanian R, Fossetta J, Tian F, Trivedi P, Lundell D, Palani A.
Xiao D, et al. Among authors: sofolarides m.
Bioorg Med Chem Lett. 2014 Aug 1;24(15):3609-13. doi: 10.1016/j.bmcl.2014.05.024. Epub 2014 May 16.
Bioorg Med Chem Lett. 2014.
PMID: 24913714
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