Discovery of 8-Membered Ring Sulfonamides as Inhibitors of Oncogenic Mutant Isocitrate Dehydrogenase 1.
Law JM, Stark SC, Liu K, Liang NE, Hussain MM, Leiendecker M, Ito D, Verho O, Stern AM, Johnston SE, Zhang YL, Dunn GP, Shamji AF, Schreiber SL.
Law JM, et al.
ACS Med Chem Lett. 2016 Aug 18;7(10):944-949. doi: 10.1021/acsmedchemlett.6b00264. eCollection 2016 Oct 13.
ACS Med Chem Lett. 2016.
PMID: 27774134
Free PMC article.