Tropmann K - Search Results

1

Abolishing Dopamine D_2long/D₃ Receptor Affinity of Subtype-Selective Carbamoylguanidine-Type Histamine H₂ Receptor Agonists.

Tropmann K, Bresinsky M, Forster L, Mönnich D, Buschauer A, Wittmann HJ, Hübner H, Gmeiner P, Pockes S, Strasser A. Tropmann K, et al. J Med Chem. 2021 Jun 24;64(12):8684-8709. doi: 10.1021/acs.jmedchem.1c00692. Epub 2021 Jun 10. J Med Chem. 2021. PMID: 34110814

2

Histamine H₂ receptor radioligands: triumphs and challenges.

Pockes S, Tropmann K. Pockes S, et al. Among authors: tropmann k. Future Med Chem. 2021 Jun;13(12):1073-1081. doi: 10.4155/fmc-2021-0058. Epub 2021 Apr 28. Future Med Chem. 2021. PMID: 33906421 Free article. Review.

3

Discovery of a G Protein-Biased Radioligand for the Histamine H₂ Receptor with Reversible Binding Properties.

Tropmann K, Höring C, Plank N, Pockes S. Tropmann K, et al. J Med Chem. 2020 Nov 12;63(21):13090-13102. doi: 10.1021/acs.jmedchem.0c01494. Epub 2020 Oct 27. J Med Chem. 2020. PMID: 33108724

4

Pharmacological characterization of a new series of carbamoylguanidines reveals potent agonism at the H₂R and D₃R.

Biselli S, Bresinsky M, Tropmann K, Forster L, Honisch C, Buschauer A, Bernhardt G, Pockes S. Biselli S, et al. Among authors: tropmann k. Eur J Med Chem. 2021 Mar 15;214:113190. doi: 10.1016/j.ejmech.2021.113190. Epub 2021 Jan 19. Eur J Med Chem. 2021. PMID: 33548637

5

Shining light on the histamine H₂ receptor: Synthesis of carbamoylguanidine-type agonists as a pharmacological tool to study internalization.

Tropmann K, Seibel-Ehlert U, Littmann T, Strasser A. Tropmann K, et al. Bioorg Med Chem Lett. 2021 Nov 15;52:128388. doi: 10.1016/j.bmcl.2021.128388. Epub 2021 Sep 30. Bioorg Med Chem Lett. 2021. PMID: 34600035

6

NanoBRET binding assay for histamine H₂ receptor ligands using live recombinant HEK293T cells.

Grätz L, Tropmann K, Bresinsky M, Müller C, Bernhardt G, Pockes S. Grätz L, et al. Among authors: tropmann k. Sci Rep. 2020 Aug 6;10(1):13288. doi: 10.1038/s41598-020-70332-3. Sci Rep. 2020. PMID: 32764682 Free PMC article.

7

A Dynamic, Split-Luciferase-Based Mini-G Protein Sensor to Functionally Characterize Ligands at All Four Histamine Receptor Subtypes.

Höring C, Seibel U, Tropmann K, Grätz L, Mönnich D, Pitzl S, Bernhardt G, Pockes S, Strasser A. Höring C, et al. Among authors: tropmann k. Int J Mol Sci. 2020 Nov 10;21(22):8440. doi: 10.3390/ijms21228440. Int J Mol Sci. 2020. PMID: 33182741 Free PMC article.

8

Author Correction: NanoBRET binding assay for histamine H₂ receptor ligands using live recombinant HEK293T cells.

Grätz L, Tropmann K, Bresinsky M, Müller C, Bernhardt G, Pockes S. Grätz L, et al. Among authors: tropmann k. Sci Rep. 2021 May 18;11(1):10747. doi: 10.1038/s41598-021-89954-2. Sci Rep. 2021. PMID: 34006951 Free PMC article. No abstract available.

9

Author Correction: NanoBRET binding assay for histamine H₂ receptor ligands using live recombinant HEK293T cells.

Grätz L, Tropmann K, Bresinsky M, Müller C, Bernhardt G, Pockes S. Grätz L, et al. Among authors: tropmann k. Sci Rep. 2021 Jun 8;11(1):12444. doi: 10.1038/s41598-021-91782-3. Sci Rep. 2021. PMID: 34103640 Free PMC article. No abstract available.

10

Fluorescent H₂ Receptor Squaramide-Type Antagonists: Synthesis, Characterization, and Applications.

Biselli S, Alencastre I, Tropmann K, Erdmann D, Chen M, Littmann T, Maia AF, Gomez-Lazaro M, Tanaka M, Ozawa T, Keller M, Lamghari M, Buschauer A, Bernhardt G. Biselli S, et al. Among authors: tropmann k. ACS Med Chem Lett. 2020 Jul 20;11(8):1521-1528. doi: 10.1021/acsmedchemlett.0c00033. eCollection 2020 Aug 13. ACS Med Chem Lett. 2020. PMID: 32832018 Free PMC article.

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