dos Santos DJ - Search Results

1

Incorporation of basic side chains into cryptolepine scaffold: structure-antimalarial activity relationships and mechanistic studies.

Lavrado J, Cabal GG, Prudêncio M, Mota MM, Gut J, Rosenthal PJ, Díaz C, Guedes RC, dos Santos DJ, Bichenkova E, Douglas KT, Moreira R, Paulo A. Lavrado J, et al. Among authors: dos santos dj. J Med Chem. 2011 Feb 10;54(3):734-50. doi: 10.1021/jm101383f. Epub 2011 Jan 5. J Med Chem. 2011. PMID: 21207937

2

Design, synthesis and structure-activity relationships of (1H-pyridin-4-ylidene)amines as potential antimalarials.

Rodrigues T, Guedes RC, dos Santos DJ, Carrasco M, Gut J, Rosenthal PJ, Moreira R, Lopes F. Rodrigues T, et al. Among authors: dos santos dj. Bioorg Med Chem Lett. 2009 Jul 1;19(13):3476-80. doi: 10.1016/j.bmcl.2009.05.017. Epub 2009 May 9. Bioorg Med Chem Lett. 2009. PMID: 19467600

3

Synthesis and evaluation of vinyl sulfones as caspase-3 inhibitors. A structure-activity study.

Newton AS, Glória PM, Gonçalves LM, dos Santos DJ, Moreira R, Guedes RC, Santos MM. Newton AS, et al. Among authors: dos santos dj, santos mm. Eur J Med Chem. 2010 Sep;45(9):3858-63. doi: 10.1016/j.ejmech.2010.05.039. Epub 2010 May 24. Eur J Med Chem. 2010. PMID: 20541849

4

Properties and behaviour of tetracyclic allopsoralen derivatives inside a DPPC lipid bilayer model.

dos Santos DJ, Saenz-Méndez P, Eriksson LA, Guedes RC. dos Santos DJ, et al. Phys Chem Chem Phys. 2011 Jun 7;13(21):10174-82. doi: 10.1039/c0cp02245d. Epub 2011 Apr 21. Phys Chem Chem Phys. 2011. PMID: 21512685

5

Toward a better pharmacophore description of P-glycoprotein modulators, based on macrocyclic diterpenes from Euphorbia species.

Ferreira RJ, dos Santos DJ, Ferreira MJ, Guedes RC. Ferreira RJ, et al. Among authors: dos santos dj. J Chem Inf Model. 2011 Jun 27;51(6):1315-24. doi: 10.1021/ci200145p. Epub 2011 Jun 9. J Chem Inf Model. 2011. PMID: 21604687

6

Identification of new antimalarial leads by use of virtual screening against cytochrome bc₁.

Rodrigues T, Moreira R, Gut J, Rosenthal PJ, O Neill PM, Biagini GA, Lopes F, dos Santos DJ, Guedes RC. Rodrigues T, et al. Among authors: dos santos dj. Bioorg Med Chem. 2011 Nov 1;19(21):6302-8. doi: 10.1016/j.bmc.2011.09.004. Epub 2011 Sep 10. Bioorg Med Chem. 2011. PMID: 21958736

7

Enhancing macrocyclic diterpenes as multidrug-resistance reversers: structure-activity studies on jolkinol D derivatives.

Reis M, Ferreira RJ, Santos MM, dos Santos DJ, Molnár J, Ferreira MJ. Reis M, et al. Among authors: dos santos dj, santos mm. J Med Chem. 2013 Feb 14;56(3):748-60. doi: 10.1021/jm301441w. Epub 2013 Jan 30. J Med Chem. 2013. PMID: 23336337

8

Synthesis, G-quadruplex stabilisation, docking studies, and effect on cancer cells of indolo[3,2-b]quinolines with one, two, or three basic side chains.

Lavrado J, Borralho PM, Ohnmacht SA, Castro RE, Rodrigues CM, Moreira R, dos Santos DJ, Neidle S, Paulo A. Lavrado J, et al. Among authors: dos santos dj. ChemMedChem. 2013 Oct;8(10):1648-61. doi: 10.1002/cmdc.201300288. Epub 2013 Aug 19. ChemMedChem. 2013. PMID: 23960016 Free article.

9

Flavones as isosteres of 4(1H)-quinolones: discovery of ligand efficient and dual stage antimalarial lead compounds.

Rodrigues T, Ressurreição AS, da Cruz FP, Albuquerque IS, Gut J, Carrasco MP, Gonçalves D, Guedes RC, dos Santos DJ, Mota MM, Rosenthal PJ, Moreira R, Prudêncio M, Lopes F. Rodrigues T, et al. Among authors: dos santos dj. Eur J Med Chem. 2013 Nov;69:872-80. doi: 10.1016/j.ejmech.2013.09.008. Epub 2013 Sep 20. Eur J Med Chem. 2013. PMID: 24125849

10

Probing the aurone scaffold against Plasmodium falciparum: design, synthesis and antimalarial activity.

Carrasco MP, Newton AS, Gonçalves L, Góis A, Machado M, Gut J, Nogueira F, Hänscheid T, Guedes RC, dos Santos DJ, Rosenthal PJ, Moreira R. Carrasco MP, et al. Among authors: dos santos dj. Eur J Med Chem. 2014 Jun 10;80:523-34. doi: 10.1016/j.ejmech.2014.04.076. Epub 2014 Apr 28. Eur J Med Chem. 2014. PMID: 24813880

Save citations to file

Email citations

Send citations to clipboard

Add to Collections

Add to My Bibliography

Create a file for external citation management software

Your saved search

Your RSS Feed

My NCBI Filters

Text availability

Article attribute

Article type

Publication date

58 results

Search Page