Digiacomo M - Search Results

1

SAR study on arylmethyloxyphenyl scaffold: looking for a P-gp nanomolar affinity.

Nesi G, Colabufo NA, Contino M, Perrone MG, Digiacomo M, Perrone R, Lapucci A, Macchia M, Rapposelli S. Nesi G, et al. Among authors: digiacomo m. Eur J Med Chem. 2014 Apr 9;76:558-66. doi: 10.1016/j.ejmech.2014.02.051. Epub 2014 Feb 21. Eur J Med Chem. 2014. PMID: 24607999

2

NO-sartans: a new class of pharmacodynamic hybrids as cardiovascular drugs.

Breschi MC, Calderone V, Digiacomo M, Martelli A, Martinotti E, Minutolo F, Rapposelli S, Balsamo A. Breschi MC, et al. Among authors: digiacomo m. J Med Chem. 2004 Nov 4;47(23):5597-600. doi: 10.1021/jm049681p. J Med Chem. 2004. PMID: 15509155

3

New NO-releasing pharmacodynamic hybrids of losartan and its active metabolite: design, synthesis, and biopharmacological properties.

Breschi MC, Calderone V, Digiacomo M, Macchia M, Martelli A, Martinotti E, Minutolo F, Rapposelli S, Rossello A, Testai L, Balsamo A. Breschi MC, et al. Among authors: digiacomo m. J Med Chem. 2006 Apr 20;49(8):2628-39. doi: 10.1021/jm0600186. J Med Chem. 2006. PMID: 16610806

4

Arylmethyloxyphenyl derivatives: small molecules displaying P-glycoprotein inhibition.

Colabufo NA, Berardi F, Perrone R, Rapposelli S, Digiacomo M, Balsamo A. Colabufo NA, et al. Among authors: digiacomo m. J Med Chem. 2006 Nov 2;49(22):6607-13. doi: 10.1021/jm060639z. J Med Chem. 2006. PMID: 17064079

5

Metabolically labile cannabinoid esters: a 'soft drug' approach for the development of cannabinoid-based therapeutic drugs.

Minutolo F, Cascio MG, Carboni I, Bisogno T, Prota G, Bertini S, Digiacomo M, Bifulco M, Di Marzo V, Macchia M. Minutolo F, et al. Among authors: digiacomo m. Bioorg Med Chem Lett. 2007 Sep 1;17(17):4878-81. doi: 10.1016/j.bmcl.2007.06.055. Epub 2007 Jun 20. Bioorg Med Chem Lett. 2007. PMID: 17604171

6

Evaluation of the NO-releasing properties of NO-donor linkers.

Calderone V, Digiacomo M, Martelli A, Minutolo F, Rapposelli S, Testai L, Balsamo A. Calderone V, et al. Among authors: digiacomo m. J Pharm Pharmacol. 2008 Feb;60(2):189-95. doi: 10.1211/jpp.60.2.0007. J Pharm Pharmacol. 2008. PMID: 18237466

7

Synthesis and biological evaluation of (hetero)arylmethyloxy- and arylmethylamine-phenyl derivatives as potent P-glycoprotein modulating agents.

Colabufo NA, Berardi F, Perrone R, Rapposelli S, Digiacomo M, Vanni M, Balsamo A. Colabufo NA, et al. Among authors: digiacomo m. J Med Chem. 2008 Mar 13;51(5):1415-22. doi: 10.1021/jm701267q. Epub 2008 Feb 8. J Med Chem. 2008. PMID: 18257545

8

alpha-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors.

Asso V, Ghilardi E, Bertini S, Digiacomo M, Granchi C, Minutolo F, Rapposelli S, Bortolato A, Moro S, Macchia M. Asso V, et al. Among authors: digiacomo m. ChemMedChem. 2008 Oct;3(10):1530-4. doi: 10.1002/cmdc.200800162. ChemMedChem. 2008. PMID: 18781572 No abstract available.

9

Spirocyclic benzopyran-based derivatives as new anti-ischemic activators of mitochondrial ATP-sensitive potassium channel.

Breschi MC, Calderone V, Digiacomo M, Manganaro M, Martelli A, Minutolo F, Rapposelli S, Testai L, Tonelli F, Balsamo A. Breschi MC, et al. Among authors: digiacomo m. J Med Chem. 2008 Nov 13;51(21):6945-54. doi: 10.1021/jm800956g. Epub 2008 Oct 17. J Med Chem. 2008. PMID: 18925735

10

2-[(3-Methoxyphenylethyl)phenoxy]-based ABCB1 inhibitors: effect of different basic side-chains on their biological properties.

Colabufo NA, Berardi F, Perrone R, Rapposelli S, Digiacomo M, Vanni M, Balsamo A. Colabufo NA, et al. Among authors: digiacomo m. J Med Chem. 2008 Dec 11;51(23):7602-13. doi: 10.1021/jm800928j. J Med Chem. 2008. PMID: 19053888

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